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kelatorphan , CAS No.92175-57-0, Inhibitor of Leukotriene A 4 hydrolase;Inhibitor of Neutral endopeptidase

  • Moligand™
Item Number
K611327
Grouped product items
SKUSizeAvailabilityPrice Qty
K611327-5mg
5mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$720.90
K611327-25mg
25mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$2,500.90
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Leukotriene A4 hydrolase Inhibitor Neutral endopeptidase Inhibitor

Basic Description

Synonymskelatorphan|92175-57-0|(3-(N-Hydroxy)carboxamido-2-benzylpropanoyl)alanine|46BBW2U5D6|n-[(2r)-2-benzyl-4-(hydroxyamino)-4-oxobutanoyl]-l-alanine|((R)-2-benzyl-4-(hydroxyamino)-4-oxobutanoyl)-L-alanine|UNII-46BBW2U5D6|3b7u|(2S)-2-[[(2R)-2-benzyl-4-(hydroxy
Specifications & PurityMoligand™
GradeMoligand™
Action TypeINHIBITOR
Mechanism of actionInhibitor of Leukotriene A 4 hydrolase;Inhibitor of Neutral endopeptidase

Associated Targets

ECE1 Tchem Endothelin-converting enzyme 1 1 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

MME Tclin Neprilysin 1 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

LTA4H Tchem Leukotriene A-4 hydrolase 4 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

ACE Tclin Angiotensin-converting enzyme 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

ANPEP Tchem Aminopeptidase N 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

Names and Identifiers

IUPAC Name (2S)-2-[[(2R)-2-benzyl-4-(hydroxyamino)-4-oxobutanoyl]amino]propanoic acid
INCHI InChI=1S/C14H18N2O5/c1-9(14(19)20)15-13(18)11(8-12(17)16-21)7-10-5-3-2-4-6-10/h2-6,9,11,21H,7-8H2,1H3,(H,15,18)(H,16,17)(H,19,20)/t9-,11+/m0/s1
InChi Key OJCFZTVYDSKXNM-GXSJLCMTSA-N
Canonical SMILES CC(C(=O)O)NC(=O)C(CC1=CC=CC=C1)CC(=O)NO
Isomeric SMILES C[C@@H](C(=O)O)NC(=O)[C@H](CC1=CC=CC=C1)CC(=O)NO
Alternate CAS 92175-57-0
PubChem CID 123982
MeSH Entry Terms (3-(N-hydroxy)carboxamido-2--benzylpropanoyl)alanine;kelatorphan

Certificates

Certificate of Analysis(COA)

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Related Documents

 SDS

 Specification Sheet

References

1. Tholander F, Roques BP, Fournié-Zaluski MC, Thunnissen MM, Haeggström JZ.  (2010)  Crystal structure of leukotriene A4 hydrolase in complex with kelatorphan, implications for design of zinc metallopeptidase inhibitors..  FEBS Lett,  584  (15): (3446-51).  [PMID:20609366]

Solution Calculators

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