| SKU | Size | Availability | Price | Qty |
|---|---|---|---|---|
| L422469-1ml | 1ml | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $241.90 |
MTP Inhibitors
| Synonyms | Lomitapide mesylate|202914-84-9|BMS 201038-04|AEGR-733 mesylate|Aegr-733 mesilate|BMS-201038-04|Lomitapide (mesylate)|lomitapide mesilate|Lomitapide mesylate [USAN]|UNII-X4S83CP54E|X4S83CP54E|lomitapide monomesylate|CHEBI:72299|lomitapide methanesulfonate |
|---|---|
| Specifications & Purity | 10mM in DMSO |
| Storage Temp | Store at -80°C |
| Shipped In | Ice chest + Ice pads |
| Product Description | Information Lomitapide Mesylate Lomitapide Mesylate is a potent microsomal triglyceride transfer protein (MTP) inhibitor, used in the treatment of familial hypercholesterolemia. |
| ALogP | 7.377 |
|---|---|
| HBD Count | 2 |
| Rotatable Bond | 12 |
| IUPAC Name | methanesulfonic acid;N-(2,2,2-trifluoroethyl)-9-[4-[4-[[2-[4-(trifluoromethyl)phenyl]benzoyl]amino]piperidin-1-yl]butyl]fluorene-9-carboxamide |
|---|---|
| INCHI | InChI=1S/C39H37F6N3O2.CH4O3S/c40-38(41,42)25-46-36(50)37(33-13-5-3-10-30(33)31-11-4-6-14-34(31)37)21-7-8-22-48-23-19-28(20-24-48)47-35(49)32-12-2-1-9-29(32)26-15-17-27(18-16-26)39(43,44)45;1-5(2,3)4/h1-6,9-18,28H,7-8,19-25H2,(H,46,50)(H,47,49);1H3,(H,2,3,4) |
| InChi Key | QKVKOFVWUHNEBX-UHFFFAOYSA-N |
| Canonical SMILES | CS(=O)(=O)O.C1CN(CCC1NC(=O)C2=CC=CC=C2C3=CC=C(C=C3)C(F)(F)F)CCCCC4(C5=CC=CC=C5C6=CC=CC=C64)C(=O)NCC(F)(F)F |
| Isomeric SMILES | CS(=O)(=O)O.C1CN(CCC1NC(=O)C2=CC=CC=C2C3=CC=C(C=C3)C(F)(F)F)CCCCC4(C5=CC=CC=C5C6=CC=CC=C64)C(=O)NCC(F)(F)F |
| PubChem CID | 11274333 |
| Molecular Weight | 789.83 |
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| DMSO(mg / mL) Max Solubility | 100 |
|---|---|
| DMSO(mM) Max Solubility | 126.6095236 |
| Water(mg / mL) Max Solubility | ＜1 |
| Pictogram(s) | GHS08 |
|---|---|
| Signal | Danger |
| Hazard Statements | H351:Suspected of causing cancer H413:May cause long lasting harmful effects to aquatic life H360:May damage fertility or the unborn child |
| Precautionary Statements | P273:Avoid release to the environment. P280:Wear protective gloves/protective clothing/eye protection/face protection. P405:Store locked up. P501:Dispose of contents/container to ... P203:Obtain, read and follow all safety instructions before use. P318:if exposed or concerned, get medical advice. |
