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MS363 , CAS No.M612086, Inhibitor of bromodomain containing 3;Inhibitor of bromodomain PHD finger transcription factor

  • Moligand™
Item Number
M612086
Grouped product items
SKUSizeAvailabilityPrice Qty
M612086-5mg
5mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$1,334.90
M612086-25mg
25mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$2,000.90
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bromodomain containing 3 Inhibitor bromodomain PHD finger transcription factor Inhibitor

Basic Description

SynonymsMS363|CHEMBL3086885|4-[(2E)-2-(2-amino-3-chloro-5-methyl-4-oxocyclohexa-2,5-dien-1-ylidene)hydrazinyl]-N-pyridin-2-ylbenzenesulfonamide|compound 29|GTPL8876|SCHEMBL12486296|SCHEMBL12486300|DTXSID101118304|BDBM50443230|PD144799|Q27087802|Cc1cc(N=Nc2ccc(cc2
Specifications & PurityMoligand™
GradeMoligand™
Action TypeINHIBITOR
Mechanism of actionInhibitor of bromodomain containing 3;Inhibitor of bromodomain PHD finger transcription factor

Associated Targets

CREBBP Tchem CREB-binding protein 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

BRD4 Tchem Bromodomain-containing protein 4 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

KAT2B Tchem Histone acetyltransferase KAT2B 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

SMARCA4 Tchem Transcription activator BRG1 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

BPTF Tchem Nucleosome-remodeling factor subunit BPTF 1 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

BRD7 Tchem Bromodomain-containing protein 7 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

BRD3 Tchem Bromodomain-containing protein 3 1 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

BAZ2B Tchem Bromodomain adjacent to zinc finger domain protein 2B 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

Names and Identifiers

IUPAC Name 4-[(2E)-2-(2-amino-3-chloro-5-methyl-4-oxocyclohexa-2,5-dien-1-ylidene)hydrazinyl]-N-pyridin-2-ylbenzenesulfonamide
INCHI InChI=1S/C18H16ClN5O3S/c1-11-10-14(17(20)16(19)18(11)25)23-22-12-5-7-13(8-6-12)28(26,27)24-15-4-2-3-9-21-15/h2-10,22H,20H2,1H3,(H,21,24)/b23-14+
InChi Key GLWPTCULLHMSCO-OEAKJJBVSA-N
Canonical SMILES NC1=C(Cl)C(=O)C(=C/C/1=N\Nc1ccc(cc1)S(=O)(=O)Nc1ccccn1)C
Isomeric SMILES CC1=CC(=C(C(=C1O)Cl)N)N=NC2=CC=C(C=C2)S(=O)(=O)NC3=CC=CC=N3
PubChem CID 136226511

Certificates

Certificate of Analysis(COA)

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Related Documents

 SDS

 Specification Sheet

References

1. Zhang G, Plotnikov AN, Rusinova E, Shen T, Morohashi K, Joshua J, Zeng L, Mujtaba S, Ohlmeyer M, Zhou MM.  (2013)  Structure-guided design of potent diazobenzene inhibitors for the BET bromodomains..  J Med Chem,  56  (22): (9251-64).  [PMID:24144283]

Solution Calculators

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