N-{3-[(5-cyclopropyl-2-{[4-(morpholin-4-yl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide , CAS No.N608785, Inhibitor of inhibitor of nuclear factor kappa B kinase subunit epsilon;Inhibitor of microtubule affinity regulating kinase 3;Inhibitor of mitogen-activated protein kinase kinase kinase 7;Inhibitor of TANK binding kinase 1
N-{3-[(5-cyclopropyl-2-{[4-(morpholin-4-yl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide , CAS No.N608785, Inhibitor of inhibitor of nuclear factor kappa B kinase subunit epsilon;Inhibitor of microtubule affinity regulating kinase 3;Inhibitor of mitogen-activated protein kinase kinase kinase 7;Inhibitor of TANK binding kinase 1
Inhibitor of inhibitor of nuclear factor kappa B kinase subunit epsilon;Inhibitor of microtubule affinity regulating kinase 3;Inhibitor of mitogen-activated protein kinase kinase kinase 7;Inhibitor of TANK binding kinase 1
1.McIver EG, Bryans J, Birchall K, Chugh J, Drake T, Lewis SJ, Osborne J, Smiljanic-Hurley E, Tsang W, Kamal A et al.. (2012) Synthesis and structure-activity relationships of a novel series of pyrimidines as potent inhibitors of TBK1/IKKε kinases.. Bioorg Med Chem Lett, 22 (23):(7169-73). [PMID:23099093]
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