Discover N,O-Didesmethyl-(rac-venlafaxine) Glucuronide Hydrochloride by Aladdin Scientific in for only $249.90. Available - in Ligands at Aladdin Scientific. a metabolite of reuptake inhibitor Venlafaxine Tags: .
Basic Description
Storage Temp
Store at -20°C
Shipped In
Ice chest + Ice pads
Product Description
N,O-Didesmethyl-(rac-venlafaxine) Glucuronide Hydrochloride is a metabolite of Venlafaxine . Venlafaxine is a derivative of phenylethylamine which is reported to facilitate neurotransmission within the central nervous system via blocking the presynaptic reuptake of neuroamines such as serotonin (5-hydroxytryptamine; 5-HT) and noradrenaline (norepinephrine). Velanfaxine is also reported to be a weak inhibitor of dopamine reuptake.|In vitro|studies indicate that Venlafaxine does not demonstrate significant activity for muscarinic, histaminergic or α-1 adrenergic receptors. The metabolism of venlafaxine is reported to occur by cytochrome P450 (CYP) enzyme CYP2D6 yielding O-desmethylvenlafaxine. A lesser metabolite, N-desmethylvenlafaxine is produced by CYP3A4.
