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norfluoxetine , CAS No.83891-03-6, Antagonist of 5-HT 2A receptor;Antagonist of 5-HT 2B receptor;Antagonist of 5-HT 2C receptor;Inhibitor of K 2P2.1;Gating inhibitor of K v3.1

Moligand™

CAS#: 83891-03-6
PubChem CID: 4541

Item Number

N612363

Grouped product items
SKU	Size	Availability	Price	Qty
N612363-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$572.90
N612363-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90

View related series

5-HT2A receptor Antagonist 5-HT2B receptor Antagonist 5-HT2C receptor Antagonist K2P2.1 Inhibitor Kv3.1 Gating inhibitor

Basic Description

Synonyms	Norfluoxetine\|83891-03-6\|Desmethylfluoxetine\|56161-73-0\|3-phenyl-3-(4-(trifluoromethyl)phenoxy)propan-1-amine\|3-phenyl-3-[4-(trifluoromethyl)phenoxy]propan-1-amine\|3-Phenyl-3-(4-trifluoromethyl-phenoxy)-propylamine\|(Phenyl-d5)\|K8D70XE2F4\|C16H16F3NO\|(R)-No
Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	ANTAGONIST, GATING INHIBITOR, INHIBITOR
Mechanism of action	Antagonist of 5-HT 2A receptor;Antagonist of 5-HT 2B receptor;Antagonist of 5-HT 2C receptor;Inhibitor of K 2P2.1;Gating inhibitor of K v3.1

Associated Targets

ABCB1 Tchem Multidrug resistance protein 1 0 Activities

Discover Target: ABCB1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

HDAC6 Tclin Histone deacetylase 6 0 Activities

Discover Target: HDAC6

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

KCNC1 Tclin Potassium voltage-gated channel subfamily C member 1 1 Activities

Discover Target: KCNC1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

CACNA1C Tclin Voltage-dependent L-type calcium channel subunit alpha-1C 1 Activities

Discover Target: CACNA1C

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

HTR2A Tclin 5-hydroxytryptamine receptor 2A 1 Activities

Discover Target: HTR2A

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

HTR2C Tclin 5-hydroxytryptamine receptor 2C 1 Activities

Discover Target: HTR2C

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

HTR2B Tclin 5-hydroxytryptamine receptor 2B 1 Activities

Discover Target: HTR2B

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

KCNK2 Tclin Potassium channel subfamily K member 2 2 Activities

Discover Target: KCNK2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

KCNH2 Tclin Potassium voltage-gated channel subfamily H member 2 1 Activities

Discover Target: KCNH2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	3-phenyl-3-[4-(trifluoromethyl)phenoxy]propan-1-amine
INCHI	InChI=1S/C16H16F3NO/c17-16(18,19)13-6-8-14(9-7-13)21-15(10-11-20)12-4-2-1-3-5-12/h1-9,15H,10-11,20H2
InChi Key	WIQRCHMSJFFONW-UHFFFAOYSA-N
Canonical SMILES	NCCC(c1ccccc1)Oc1ccc(cc1)C(F)(F)F
Isomeric SMILES	C1=CC=C(C=C1)C(CCN)OC2=CC=C(C=C2)C(F)(F)F
PubChem CID	4541

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