Determine the necessary mass, volume, or concentration for preparing a solution.
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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O275137-5mg | 5mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $68.90 | |
O275137-10mg | 10mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $115.90 | |
O275137-25mg | 25mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $224.90 | |
O275137-50mg | 50mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $406.90 | |
O275137-100mg | 100mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $607.90 |
Potent, reversible phospholipase A 2 (PLA 2 ) inhibitor
Synonyms | Ono-RS-082|99754-06-0|2-(4-amylcinnamoyl)amino-4-chlorobenzoic acid|2-(p-AMYLCINNAMOYL)AMINO-4-CHLOROBENZOIC ACID|(E)-4-CHLORO-2-(3-(4-PENTYLPHENYL)ACRYLAMIDO)BENZOIC ACID|4-chloro-2-[[(E)-3-(4-pentylphenyl)prop-2-enoyl]amino]benzoic acid|CHEMBL3818672|4- |
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Specifications & Purity | ≥98% |
Biochemical and Physiological Mechanisms | Potent, reversible PLA 2 inhibitor (IC 50 = 7 µM). Cell-permeable. Active in ex vivo preparations. |
Storage Temp | Protected from light,Store at -20°C,Desiccated |
Shipped In | Ice chest + Ice pads |
Note | Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details. |
Product Description | Store at -20°C. It is important to note that this product is reported to be light sensitive. Store In the Dark. Store under desiccating conditions. |
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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IUPAC Name | 4-chloro-2-[[(E)-3-(4-pentylphenyl)prop-2-enoyl]amino]benzoic acid |
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INCHI | InChI=1S/C21H22ClNO3/c1-2-3-4-5-15-6-8-16(9-7-15)10-13-20(24)23-19-14-17(22)11-12-18(19)21(25)26/h6-14H,2-5H2,1H3,(H,23,24)(H,25,26)/b13-10+ |
InChi Key | MDVFITMPFHDRBZ-JLHYYAGUSA-N |
Canonical SMILES | CCCCCC1=CC=C(C=C1)C=CC(=O)NC2=C(C=CC(=C2)Cl)C(=O)O |
Isomeric SMILES | CCCCCC1=CC=C(C=C1)/C=C/C(=O)NC2=C(C=CC(=C2)Cl)C(=O)O |
PubChem CID | 6438389 |
Molecular Weight | 371.9 |
Enter Lot Number to search for COA:
To view the certificate results,please click on a Lot number.For Lot numbers from past orders,please use our order status section
Lot Number | Certificate Type | Date | Item |
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H2426305 | Certificate of Analysis | May 14, 2024 | O275137 |
H2426308 | Certificate of Analysis | May 14, 2024 | O275137 |
H2426309 | Certificate of Analysis | May 14, 2024 | O275137 |
H2426337 | Certificate of Analysis | May 14, 2024 | O275137 |
H2426338 | Certificate of Analysis | May 14, 2024 | O275137 |
H2426339 | Certificate of Analysis | May 14, 2024 | O275137 |
H2426340 | Certificate of Analysis | May 14, 2024 | O275137 |
H2426341 | Certificate of Analysis | May 14, 2024 | O275137 |
H2426485 | Certificate of Analysis | May 14, 2024 | O275137 |
Solubility | Soluble in DMSO to 50 mM (with warming) and in ethanol to 25 mM (with warming) |
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Sensitivity | light sensitive |