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PD 173212 - ≥99%, high purity , CAS No.217171-01-2

  • ≥99%
Item Number
P274793
Grouped product items
SKUSizeAvailabilityPrice Qty
P274793-5mg
5mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$212.90
P274793-10mg
10mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$313.90
P274793-25mg
25mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$196.90
P274793-50mg
50mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$314.90

Potent, selective N-type voltage-gated Ca 2+ channel blocker

View related series
Calcium Channel

Basic Description

Synonyms217171-01-2|PD 173212|PD173212|Z7UUP5FPKC|PD-173212|UNII-Z7UUP5FPKC|CHEMBL299749|(2S)-N-[(2S)-1-(tert-butylamino)-1-oxo-3-(4-phenylmethoxyphenyl)propan-2-yl]-2-[(4-tert-butylphenyl)methyl-methylamino]-4-methylpentanamide|L-Tyrosinamide, N-((4-(1,1-dimethy
Specifications & Purity≥99%
Storage TempStore at -20°C,Argon charged,Desiccated
Shipped InDry ice

Associated Targets

CACNA1B Tclin Voltage-dependent N-type calcium channel subunit alpha-1B 1 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

Names and Identifiers

IUPAC Name (2S)-N-[(2S)-1-(tert-butylamino)-1-oxo-3-(4-phenylmethoxyphenyl)propan-2-yl]-2-[(4-tert-butylphenyl)methyl-methylamino]-4-methylpentanamide
INCHI InChI=1S/C38H53N3O3/c1-27(2)23-34(41(9)25-29-15-19-31(20-16-29)37(3,4)5)36(43)39-33(35(42)40-38(6,7)8)24-28-17-21-32(22-18-28)44-26-30-13-11-10-12-14-30/h10-22,27,33-34H,23-26H2,1-9H3,(H,39,43)(H,40,42)/t33-,34-/m0/s1
InChi Key GCDHMGROXQUFNR-HEVIKAOCSA-N
Canonical SMILES CC(C)CC(C(=O)NC(CC1=CC=C(C=C1)OCC2=CC=CC=C2)C(=O)NC(C)(C)C)N(C)CC3=CC=C(C=C3)C(C)(C)C
Isomeric SMILES CC(C)C[C@@H](C(=O)N[C@@H](CC1=CC=C(C=C1)OCC2=CC=CC=C2)C(=O)NC(C)(C)C)N(C)CC3=CC=C(C=C3)C(C)(C)C
PubChem CID 9916734
Molecular Weight 599.85

Certificates

Certificate of Analysis(COA)

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8 results found

Lot NumberCertificate TypeDateItem
G2417564Certificate of AnalysisApr 01, 2024 P274793
G2417581Certificate of AnalysisApr 01, 2024 P274793
G2417582Certificate of AnalysisApr 01, 2024 P274793
G2417583Certificate of AnalysisApr 01, 2024 P274793
G2417584Certificate of AnalysisApr 01, 2024 P274793
G2417623Certificate of AnalysisApr 01, 2024 P274793
G2417624Certificate of AnalysisApr 01, 2024 P274793
G2417625Certificate of AnalysisApr 01, 2024 P274793

Chemical and Physical Properties

SolubilitySoluble in DMSO to 100 mM and in ethanol to 100 mM
SensitivityMoisture sensitive

Related Documents

References

1. Okada T et al..  (2021)  Pain induces stable, active microcircuits in the somatosensory cortex that provide a therapeutic target..  Sci Adv,  (12):   [PMID:33741588]

Solution Calculators