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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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P274793-5mg | 5mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $212.90 | |
P274793-10mg | 10mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $313.90 | |
P274793-25mg | 25mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $196.90 | |
P274793-50mg | 50mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $314.90 |
Potent, selective N-type voltage-gated Ca 2+ channel blocker
Synonyms | 217171-01-2|PD 173212|PD173212|Z7UUP5FPKC|PD-173212|UNII-Z7UUP5FPKC|CHEMBL299749|(2S)-N-[(2S)-1-(tert-butylamino)-1-oxo-3-(4-phenylmethoxyphenyl)propan-2-yl]-2-[(4-tert-butylphenyl)methyl-methylamino]-4-methylpentanamide|L-Tyrosinamide, N-((4-(1,1-dimethy |
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Specifications & Purity | ≥99% |
Storage Temp | Store at -20°C,Argon charged,Desiccated |
Shipped In | Dry ice |
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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IUPAC Name | (2S)-N-[(2S)-1-(tert-butylamino)-1-oxo-3-(4-phenylmethoxyphenyl)propan-2-yl]-2-[(4-tert-butylphenyl)methyl-methylamino]-4-methylpentanamide |
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INCHI | InChI=1S/C38H53N3O3/c1-27(2)23-34(41(9)25-29-15-19-31(20-16-29)37(3,4)5)36(43)39-33(35(42)40-38(6,7)8)24-28-17-21-32(22-18-28)44-26-30-13-11-10-12-14-30/h10-22,27,33-34H,23-26H2,1-9H3,(H,39,43)(H,40,42)/t33-,34-/m0/s1 |
InChi Key | GCDHMGROXQUFNR-HEVIKAOCSA-N |
Canonical SMILES | CC(C)CC(C(=O)NC(CC1=CC=C(C=C1)OCC2=CC=CC=C2)C(=O)NC(C)(C)C)N(C)CC3=CC=C(C=C3)C(C)(C)C |
Isomeric SMILES | CC(C)C[C@@H](C(=O)N[C@@H](CC1=CC=C(C=C1)OCC2=CC=CC=C2)C(=O)NC(C)(C)C)N(C)CC3=CC=C(C=C3)C(C)(C)C |
PubChem CID | 9916734 |
Molecular Weight | 599.85 |
Enter Lot Number to search for COA:
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Lot Number | Certificate Type | Date | Item |
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G2417564 | Certificate of Analysis | Apr 01, 2024 | P274793 |
G2417581 | Certificate of Analysis | Apr 01, 2024 | P274793 |
G2417582 | Certificate of Analysis | Apr 01, 2024 | P274793 |
G2417583 | Certificate of Analysis | Apr 01, 2024 | P274793 |
G2417584 | Certificate of Analysis | Apr 01, 2024 | P274793 |
G2417623 | Certificate of Analysis | Apr 01, 2024 | P274793 |
G2417624 | Certificate of Analysis | Apr 01, 2024 | P274793 |
G2417625 | Certificate of Analysis | Apr 01, 2024 | P274793 |
Solubility | Soluble in DMSO to 100 mM and in ethanol to 100 mM |
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Sensitivity | Moisture sensitive |
1. Okada T et al.. (2021) Pain induces stable, active microcircuits in the somatosensory cortex that provide a therapeutic target.. Sci Adv, 7 (12): [PMID:33741588] |