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Transmembrane Transporters
Voltage-gated ion channels
Potassium channels
PF‐06526290 , CAS No.P612740, Gating inhibitor of Na v1.3;Gating inhibitor of Na v1.7

PF‐06526290 , CAS No.P612740, Gating inhibitor of Na v1.3;Gating inhibitor of Na v1.7

Item Number

P612740

Grouped product items
SKU	Size	Availability	Price	Qty
P612740-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,000.90
P612740-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90

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Basic Description

Synonyms	PF06526290
Grade	Moligand™
Action Type	GATING INHIBITOR
Mechanism of action	Gating inhibitor of Na v1.3;Gating inhibitor of Na v1.7

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

IUPAC Name	1-{4-[benzyl(methyl)sulfamoyl]phenyl}-3-(1,3-thiazol-2-yl)urea
INCHI	InChI=1S/C18H18N4O3S2/c1-22(13-14-5-3-2-4-6-14)27(24,25)16-9-7-15(8-10-16)20-17(23)21-18-19-11-12-26-18/h2-12H,13H2,1H3,(H2,19,20,21,23)
InChi Key	NZXOWNNCAZTBDJ-UHFFFAOYSA-N
Canonical SMILES	O=C(Nc1nccs1)Nc1ccc(cc1)S(=O)(=O)N(Cc1ccccc1)C
PubChem CID	134611890

PubChem CID	134611890

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