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PF 750 - ≥98%(HPLC), high purity , CAS No.959151-50-9, Inhibitor of epoxide hydrolase 2;Inhibitor of Fatty acid amide hydrolase

Moligand™
≥98%(HPLC)

CAS#: 959151-50-9
Formula: C₂₂H₂₃N₃O
Molecular Weight: 345.44
PubChem CID: 25154868

Item Number

P288561

Grouped product items
SKU	Size	Availability	Price
P288561-5mg	5mg	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$88.90
P288561-10mg	10mg	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$137.90
P288561-25mg	25mg	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$296.90
P288561-50mg	50mg	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$474.90
P288561-100mg	100mg	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$855.90

Selective FAAH inhibitor

View related series

epoxide hydrolase 2 Inhibitor Fatty acid amide hydrolase Inhibitor

Basic Description

Synonyms	PF 750\|959151-50-9\|PF-750\|N-phenyl-4-(quinolin-3-ylmethyl)piperidine-1-carboxamide\|1-Piperidinecarboxamide, N-phenyl-4-(3-quinolinylmethyl)-\|7756CPP14K\|N-Phenyl-4-(3-quinolinylmethyl)-1-piperidinecarboxamide\|UNII-7756CPP14K\|PF750\|CHEMBL560590\|GTPL5244\|BDB
Specifications & Purity	Moligand™, ≥98%(HPLC)
Biochemical and Physiological Mechanisms	Irreversible fatty acid amide hydrolase (FAAH) inhibitor (IC50= 16.2 nM) that displays no activity at a range of other serine hydrolases. Selectively inhibits FAAH within the central nervous system. Orally active.
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads
Grade	Moligand™
Action Type	INHIBITOR
Mechanism of action	Inhibitor of epoxide hydrolase 2;Inhibitor of Fatty acid amide hydrolase
Product Description	Product Describtion: PF 750 is a selective and covalent fatty acid amide hydrolase inhibitor, It shows IC50s varied from 16.2-595 nM in different pre-incubation times.

Associated Targets

EPHX2 Tchem Bifunctional epoxide hydrolase 2 2 Activities

Discover Target: EPHX2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

HDAC6 Tclin Histone deacetylase 6 0 Activities

Discover Target: HDAC6

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

FAAH Tchem Fatty-acid amide hydrolase 1 7 Activities

Discover Target: FAAH

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	N-phenyl-4-(quinolin-3-ylmethyl)piperidine-1-carboxamide
INCHI	InChI=1S/C22H23N3O/c26-22(24-20-7-2-1-3-8-20)25-12-10-17(11-13-25)14-18-15-19-6-4-5-9-21(19)23-16-18/h1-9,15-17H,10-14H2,(H,24,26)
InChi Key	BIODYGOZWZNCAG-UHFFFAOYSA-N
Canonical SMILES	C1CN(CCC1CC2=CC3=CC=CC=C3N=C2)C(=O)NC4=CC=CC=C4
Isomeric SMILES	C1CN(CCC1CC2=CC3=CC=CC=C3N=C2)C(=O)NC4=CC=CC=C4
WGK Germany	3
PubChem CID	25154868
Molecular Weight	345.44

CAS Registry No.

959151-50-9

PubChem CID

25154868

ChEMBL Ligand

CHEMBL560590

Certificates

Certificate of Analysis(COA)

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5 results found

Lot Number	Certificate Type	Date	Item
I2205104	Certificate of Analysis	Jun 27, 2022	P288561
I2205105	Certificate of Analysis	Jun 27, 2022	P288561
I2205106	Certificate of Analysis	Jun 27, 2022	P288561
I2205107	Certificate of Analysis	Jun 27, 2022	P288561
I2205172	Certificate of Analysis	Jun 27, 2022	P288561

Safety and Hazards(GHS)

Pictogram(s)	GHS07
Signal	Warning
Hazard Statements	H302:Harmful if swallowed
Precautionary Statements	P501:Dispose of contents/container to ... P264:Wash hands [and …] thoroughly after handling. P270:Do not eat, drink or smoke when using this product. P330:Rinse mouth. P301+P317:IF SWALLOWED: Get medical help.
WGK Germany	3
RIDADR	NONHforallmodesoftransport

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