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PQA-18 , CAS No.P612908, Inhibitor of p21 (RAC1) activated kinase 2

Item Number

P612908

Grouped product items
SKU	Size	Availability	Price	Qty
P612908-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$922.90
P612908-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$3,226.90

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Basic Description

Grade	Moligand™
Action Type	INHIBITOR
Mechanism of action	Inhibitor of p21 (RAC1) activated kinase 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

IUPAC Name	3-methylbut-2-enyl 4-methoxy-8-(3-methylbut-2-enoxy)quinoline-2-carboxylate
INCHI	InChI=1S/C25H31NO4/c1-17(2)10-13-28-22-9-7-8-20-23(29-14-11-18(3)4)16-21(26-24(20)22)25(27)30-15-12-19(5)6/h7-12,16H,13-15H2,1-6H3
InChi Key	APPXFGJVXDYNBO-UHFFFAOYSA-N
Canonical SMILES	CC(=CCOc1cc(nc2c1cccc2OCC=C(C)C)C(=O)OCC=C(C)C)C
Isomeric SMILES	CC(=CCOC1=CC=CC2=C1N=C(C=C2OC)C(=O)OCC=C(C)C)C
PubChem CID	46910769

PubChem CID	46910769
ChEMBL Ligand	CHEMBL3355920

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1. Ogura M, Kikuchi H, Suzuki T, Yamaki J, Homma MK, Oshima Y, Homma Y. (2016) Prenylated quinolinecarboxylic acid derivative suppresses immune response through inhibition of PAK2.. Biochem Pharmacol, 105 (3): (55-65). [PMID:26827943]

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