Progabide - ≥98%, high purity , CAS No.62666-20-0

Item Number

P347299

Grouped product items
SKU	Size	Availability	Price
P347299-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$44.90
P347299-10mg	10mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$76.90
P347299-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$154.90
P347299-50mg	50mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$249.90
P347299-100mg	100mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$392.90

a GABAA and GABAB receptor agonistic

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Basic Description

Synonyms	Progabide\|62666-20-0\|Halogabide\|Gabren\|Gabrene\|Progabidum [INN-Latin]\|Progabida [INN-Spanish]\|4-(((4-Chlorophenyl)(5-fluoro-2-hydroxyphenyl)methylene)amino)butanamide\|SL 76002\|Progabide, (Z)-\|SL-76002\|SL 76 002\|112E50TORV\|4-[[(E)-(4-chlorophenyl)-(3-fluor
Specifications & Purity	≥98%
Storage Temp	Store at 2-8°C
Shipped In	Ice chest + Ice pads
Product Description	Progabide is an analog and prodrug of gamma-aminobutyric acid. It has potential uses in the treatment of epilepsy. It has agonistic activity for both the GABAA and GABAB receptors.

pKa

pKa: 10.33 (Predicted)

Ki Data

GABA-A receptor; anion channel: Ki= 14 μM (rat); GABA-A receptor; anion channel: Ki= 40 μM (human)

Names and Identifiers

IUPAC Name	4-[[(4-chlorophenyl)-(5-fluoro-2-hydroxyphenyl)methylidene]amino]butanamide
INCHI	InChI=1S/C17H16ClFN2O2/c18-12-5-3-11(4-6-12)17(21-9-1-2-16(20)23)14-10-13(19)7-8-15(14)22/h3-8,10,22H,1-2,9H2,(H2,20,23)
InChi Key	IBALRBWGSVJPAP-UHFFFAOYSA-N
Canonical SMILES	C1=CC(=CC=C1C(=NCCCC(=O)N)C2=C(C=CC(=C2)F)O)Cl
Isomeric SMILES	C1=CC(=CC=C1C(=NCCCC(=O)N)C2=C(C=CC(=C2)F)O)Cl
PubChem CID	44115
Molecular Weight	334.77

Solubility

Soluble in chloroform, DMSO, and methanol.

Refractive Index

n20D1.61 (Predicted)

Boil Point(°C)

~558.1° C at 760 mmHg (Predicted)

Melt Point(°C)

135-137° C

Solution Calculators

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Basic Description