PROTAC BRD4 Degrader-9 - 98%, high purity , CAS No.2417370-42-2

  • ≥98%
Item Number
P648843
Grouped product items
SKUSizeAvailabilityPrice Qty
P648843-1mg
1mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$1,100.90
P648843-5mg
5mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$2,950.90

Basic Description

Specifications & Purity98%
Storage TempStore at -20°C
Shipped InIce chest + Ice pads
Product Description

PROTAC BRD4 Degrader-9 (compound 8a) is a PROTAC connected by ligands for von Hippel-Lindau and BRD4 . PROTAC BRD4 Degrader-9 can be conjugated with STEAP1 and CLL1 antibodies to degrade the BRD4 protein in PC3 prostate cancer cells, with a DC 50 of 0.86 nM and 7.6 nM, respectively

Form:Solid

IC50& Target:BRD4

Names and Identifiers

Canonical SMILES CC(N=CS1)=C1C2=CC=C(CNC([C@@H]3C[C@H](CN3C([C@@H](NC(COCCOCCOCCNC(C4=CC(N(C5=NC=C(F)C=C5F)CC6=CNC7=C6C8=CN(C)C7=O)=C8C=C4CS(=O)(C)=O)=O)=O)C(C)(C)C)=O)OC(OCC(C)(C)SS(C)(=O)=O)=O)=O)C=C2
Molecular Weight 1312.50

Certificates

Certificate of Analysis(COA)

Enter Lot Number to search for COA:

Related Documents

Solution Calculators