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PROTAC BRD4 Degrader-9 - 98%, high purity , CAS No.2417370-42-2

≥98%

CAS#: 2417370-42-2
Formula: C₅₉H₇₁F₂N₉O₁₅S₄
Molecular Weight: 1312.50

Item Number

P648843

Grouped product items
SKU	Size	Availability	Price	Qty
P648843-1mg	1mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,100.90
P648843-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,950.90

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Basic Description

Specifications & Purity	≥98%
Biochemical and Physiological Mechanisms	PROTAC BRD4 Degrader-9 (compound 8a) is a PROTAC connected by ligands for von Hippel-Lindau and BRD4 . PROTAC BRD4 Degrader-9 can be conjugated with STEAP1 and CLL1 antibodies to degrade the BRD4 protein in PC3 prostate cancer cells, with a DC 50 of 0.86
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads
Product Description	PROTAC BRD4 Degrader-9 (compound 8a) is a PROTAC connected by ligands for von Hippel-Lindau and BRD4 . PROTAC BRD4 Degrader-9 can be conjugated with STEAP1 and CLL1 antibodies to degrade the BRD4 protein in PC3 prostate cancer cells, with a DC 50 of 0.86 nM and 7.6 nM, respectively Form:Solid IC50& Target:BRD4

Canonical SMILES

CC(N=CS1)=C1C2=CC=C(CNC([C@@H]3C[C@H](CN3C([C@@H](NC(COCCOCCOCCNC(C4=CC(N(C5=NC=C(F)C=C5F)CC6=CNC7=C6C8=CN(C)C7=O)=C8C=C4CS(=O)(C)=O)=O)=O)C(C)(C)C)=O)OC(OCC(C)(C)SS(C)(=O)=O)=O)=O)C=C2

Molecular Weight

1312.50

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PROTAC BRD4 Degrader-9 - 98%, high purity , CAS No.2417370-42-2

Basic Description

Names and Identifiers

Certificates

Certificate of Analysis(COA)

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