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Ligand-gated ion channels
P2X receptors
PSB-12054 , CAS No.1407632-07-8, Antagonist of P2X4

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PSB-12054 , CAS No.1407632-07-8, Antagonist of P2X4

Moligand™

CAS#: 1407632-07-8
Formula: C₂₀H₁₅NO₃
Molecular Weight: 317.3
PubChem CID: 60168729

Item Number

P612986

Grouped product items
SKU	Size	Availability	Price	Qty
P612986-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,334.90
P612986-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,001.90

View related series

P2X4 Antagonist

Basic Description

Synonyms	PSB12054
Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	ANTAGONIST
Mechanism of action	Antagonist of P2X4

Associated Targets

P2RX3 Tclin P2X purinoceptor 3 1 Activities

Discover Target: P2RX3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

P2RX4 Tchem P2X purinoceptor 4 2 Activities

Discover Target: P2RX4

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

P2RX7 Tchem P2X purinoceptor 7 0 Activities

Discover Target: P2RX7

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

P2RX2 Tchem P2X purinoceptor 2 0 Activities

Discover Target: P2RX2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

P2RX1 Tchem P2X purinoceptor 1 1 Activities

Discover Target: P2RX1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	benzyl phenoxazine-10-carboxylate
INCHI	InChI=1S/C20H15NO3/c22-20(23-14-15-8-2-1-3-9-15)21-16-10-4-6-12-18(16)24-19-13-7-5-11-17(19)21/h1-13H,14H2
InChi Key	KGVCOYMLGBNCDW-UHFFFAOYSA-N
Canonical SMILES	C1=CC=C(C=C1)COC(=O)N2C3=CC=CC=C3OC4=CC=CC=C42
Isomeric SMILES	C1=CC=C(C=C1)COC(=O)N2C3=CC=CC=C3OC4=CC=CC=C42
PubChem CID	60168729
MeSH Entry Terms	N-(benzyloxycarbonyl)phenoxazine;PSB-12054
Molecular Weight	317.3

Database links

PubChem CID	60168729
CAS Registry No.	1407632-07-8
ChEMBL Ligand	CHEMBL2180137
BindingDB Ligand	50399165

Certificates

Certificate of Analysis(COA)

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References

1. Hernandez-Olmos V, Abdelrahman A, El-Tayeb A, Freudendahl D, Weinhausen S, Müller CE. (2012) N-substituted phenoxazine and acridone derivatives: structure-activity relationships of potent P2X4 receptor antagonists.. J Med Chem, 55 (22): (9576-88). [PMID:23075067]

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