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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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P347546-10mg | 10mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $127.90 | |
P347546-50mg | 50mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $395.90 |
an agonist of the GPR119 receptor
Synonyms | 388575-52-8|PSN 375963|PSN375963|PSN-375963|4-[5-(4-butylcyclohexyl)-1,2,4-oxadiazol-3-yl]pyridine|PSN-375,963|SCHEMBL385375|GTPL3318|CHEMBL4303425|5-(4-butylcyclohexyl)-3-pyridin-4-yl-1,2,4-oxadiazole|C9M28M425E|DTXSID201028459|HMS3650E12|AKOS040745320|N |
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Specifications & Purity | Moligand™, ≥98% |
Storage Temp | Room temperature,Desiccated |
Shipped In | Normal |
Grade | Moligand™ |
Action Type | AGONIST |
Mechanism of action | Agonist of GPR119 |
Product Description | PSN 375963 hydrochloride is a GPR119 receptor agonist (EC50 values are 8.4 and 7.9 μM at human and mouse receptors respectively). Displays similar potency to the endogenous ligand oleylethanolamide (OEA). |
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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IUPAC Name | 5-(4-butylcyclohexyl)-3-pyridin-4-yl-1,2,4-oxadiazole |
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INCHI | InChI=1S/C17H23N3O/c1-2-3-4-13-5-7-15(8-6-13)17-19-16(20-21-17)14-9-11-18-12-10-14/h9-13,15H,2-8H2,1H3 |
InChi Key | OAVLEYPTWABFLF-UHFFFAOYSA-N |
Canonical SMILES | CCCCC1CCC(CC1)C2=NC(=NO2)C3=CC=NC=C3 |
Isomeric SMILES | CCCCC1CCC(CC1)C2=NC(=NO2)C3=CC=NC=C3 |
PubChem CID | 2875918 |
Molecular Weight | 285.38 |
CAS Registry No. | 388575-52-8 |
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Wikipedia | PSN375963 |
PubChem CID | 2875918 |
GPCRdb Ligand | PSN375963 |
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Solubility | Soluble in ethanol (100 mM), and DMSO (100 mM). |
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Refractive Index | n20D1.52 (Predicted) |
RIDADR | NONHforallmodesoftransport |
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