Discover R-Venlafaxine-di-p-toluoyl-D-tartrate Salt by Aladdin Scientific in for only $581.90. Available - in Ligands at Aladdin Scientific. a (?)-Venlafaxine derivative Tags: .
Basic Description
Synonyms
SCHEMBL4310168 | (2S,3S)-2,3-bis[(4-methylbenzoyl)oxy]butanedioic acid;1-[(1R)-2-(dimethylamino)-1-(4-methoxyphenyl)ethyl]cyclohexan-1-ol | R-Venlafaxine Di-p-toluoyl-D-tartrate Salt | J-016718 | DTXSID60476505 | R-Venlafaxine-di-p-toluoyl-D-tartrate Salt
Storage Temp
Store at -20°C
Shipped In
Ice chest + Ice pads
Product Description
R-Venlafaxine-di-p-toluoyl-D-tartrate Salt is a derivative of (-)-Venlafaxine. Venlafaxine is a derivative of phenylethylamine which is reported to facilitate neurotransmission within the central nervous system via blocking the presynaptic reuptake of neuroamines such as serotonin (5-hydroxytryptamine; 5-HT) and noradrenaline (norepinephrine). Venlafaxine is also reported to be a weak inhibitor of dopamine reuptake.|In vitro|studies indicate that Venlafaxine does not demonstrate significant activity for muscarinic, histaminergic or α-1 adrenergic receptors. The metabolism of venlafaxine is reported to occur by cytochrome P450 (CYP) enzyme CYP2D6 yielding O-desmethylvenlafaxine. A lesser metabolite, N-desmethylvenlafaxine is produced by CYP3A4.