Sepimostat - 98%, high purity , CAS No.103926-64-3

Item Number

S413390

Grouped product items
SKU	Size	Availability	Price
S413390-1mg	1mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$92.90
S413390-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$296.90
S413390-10mg	10mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$399.90
S413390-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$939.90
S413390-50mg	50mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$949.90
S413390-100mg	100mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,299.90

View related series

Basic Description

Synonyms	SCHEMBL15535526 \| Sepimostat [INN] \| CS-0127905 \| Q27263101 \| HY-136299 \| F81697 \| (6-carbamimidoylnaphthalen-2-yl) 4-(4,5-dihydro-1H-imidazol-2-ylamino)benzoate \| UNII-5ZFR16F4QQ \| Sepimostat \| 6-Carbamimidoylnaphthalen-2-yl 4-((4,5-dihydro-1H-imidazol-2
Specifications & Purity	≥98%
Biochemical and Physiological Mechanisms	Sepimostat (FUT-187 free base) is an inhibitor of Ifenprodil binding with Ki of 27.7\u2009 μM. Sepimostat is an antagonist of NR2B N-methyl-D-aspartate receptor acting at the Ifenprodil-binding site of the NR2B subunit with neuroprotective activity.
Storage Temp	Protected from light,Store at -20°C,Argon charged
Shipped In	Ice chest + Ice pads
Product Description	Information Sepimostat (FUT-187 free base) is an inhibitor of Ifenprodil binding with Ki of 27.7 μM. Sepimostat is an antagonist of NR2B N-methyl-D-aspartate receptor acting at the Ifenprodil-binding site of the NR2B subunit with neuroprotective activity.

Associated Targets

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	(6-carbamimidoylnaphthalen-2-yl) 4-(4,5-dihydro-1H-imidazol-2-ylamino)benzoate
INCHI	InChI=1S/C21H19N5O2/c22-19(23)16-2-1-15-12-18(8-5-14(15)11-16)28-20(27)13-3-6-17(7-4-13)26-21-24-9-10-25-21/h1-8,11-12H,9-10H2,(H3,22,23)(H2,24,25,26)
InChi Key	QMRJOIUGPCVZPH-UHFFFAOYSA-N
Canonical SMILES	C1CN=C(N1)NC2=CC=C(C=C2)C(=O)OC3=CC4=C(C=C3)C=C(C=C4)C(=N)N
Isomeric SMILES	C1CN=C(N1)NC2=CC=C(C=C2)C(=O)OC3=CC4=C(C=C3)C=C(C=C4)C(=N)N
PubChem CID	108041
Molecular Weight	373.4

Safety and Hazards(GHS)

Signal	Warning
Hazard Statements	H315:Causes skin irritation H319:Causes serious eye irritation H335:May cause respiratory irritation H302:Harmful if swallowed
Precautionary Statements	P261:Avoid breathing dust/fume/gas/mist/vapors/spray. P305+P351+P338:IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses if present and easy to do - continue rinsing. P280:Wear protective gloves/protective clothing/eye protection/face protection. P302+P352:IF ON SKIN: wash with plenty of water. P301+P312:IF SWALLOWED: call a POISON CENTER/doctor/... IF you feel unwell.

Solution Calculators

Determine the necessary mass, volume, or concentration for preparing a solution.

Determine the dilution needed to prepare a stock solution.

Basic Description