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SGC GAK 1 - 98%, high purity , CAS No.2226517-76-4

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SGC GAK 1 - 98%, high purity , CAS No.2226517-76-4

≥98%

CAS#: 2226517-76-4
Formula: C₁₈H₁₇BrN₂O₃
Molecular Weight: 389.24
PubChem CID: 134812846

Item Number

S288622

Grouped product items
SKU	Size	Availability	Price
S288622-5mg	5mg	In stock	$88.90
S288622-10mg	10mg	In stock	$147.90
S288622-25mg	25mg	In stock	$296.90
S288622-50mg	50mg	In stock	$474.90
S288622-100mg	100mg	In stock	$751.90

High affinity cyclin G associated kinase (GAK) inhibitor

Basic Description

Synonyms	SGC-GAK-1;6-bromo-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine;6-Bromo-N-(3,4,5-trimethoxyphenyl)-4-quinolinamine
Specifications & Purity	98%
Storage Temp	Store at -20°C
Shipped In	Dry ice

Associated Targets

GAK Tchem Cyclin-G-associated kinase 4 Activities

Discover Target: GAK

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	6-bromo-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine
INCHI	InChI=1S/C18H17BrN2O3/c1-22-16-9-12(10-17(23-2)18(16)24-3)21-15-6-7-20-14-5-4-11(19)8-13(14)15/h4-10H,1-3H3,(H,20,21)
InChi Key	AUOSKLDNVNGKRR-UHFFFAOYSA-N
Canonical SMILES	COC1=CC(=CC(=C1OC)OC)NC2=C3C=C(C=CC3=NC=C2)Br
Isomeric SMILES	COC1=CC(=CC(=C1OC)OC)NC2=C3C=C(C=CC3=NC=C2)Br
PubChem CID	134812846
Molecular Weight	389.24

Certificates

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5 results found

Lot Number	Certificate Type	Date	Item
K2101138	Certificate of Analysis	Aug 19, 2024	S288622
K2101139	Certificate of Analysis	Aug 19, 2024	S288622
K2101140	Certificate of Analysis	Aug 19, 2024	S288622
K2101141	Certificate of Analysis	Aug 19, 2024	S288622
K2101142	Certificate of Analysis	Aug 19, 2024	S288622

Chemical and Physical Properties

Solubility	Soluble in DMSO, the highest concentration (mg/mL): 78, the highest concentration (mM): 200.39；; Soluble in ethanol, the highest concentration (mg/mL): 39, the highest concentration (mM): 100.2；; Insoluble in water

Safety and Hazards(GHS)

Pictogram(s)	GHS07
Signal	Warning
Hazard Statements	H315:Causes skin irritation H319:Causes serious eye irritation H335:May cause respiratory irritation H302:Harmful if swallowed
Precautionary Statements	P261:Avoid breathing dust/fume/gas/mist/vapors/spray. P305+P351+P338:IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses if present and easy to do - continue rinsing.

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