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Sigma-1 receptor antagonist 3 - 10mM in DMSO, high purity , CAS No.1639220-17-9(DMSO)

Sigma-1 receptor antagonist 3 - 10mM in DMSO, high purity , CAS No.1639220-17-9(DMSO)

Item Number

S655395

Grouped product items
SKU	Size	Availability	Price	Qty
S655395-1ml	1ml	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$330.90

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Basic Description

Specifications & Purity	10mM in DMSO
Storage Temp	Store at -80°C
Shipped In	Ice chest + Ice pads
Product Description	Sigma-1 receptor antagonist 3 (compound135) is a potent and selective Sigma-1 (σ1) receptor antagonist with a K i of 1.14 nM. Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG) with an IC 50 of 1.54 μM. Sigma-1 receptor antagonist 3 has the potential for the neuropathic pain IC50& Target:IC50: 1.54μM (hERG),Ki : 1.14 nM (Sigma-1 receptor),1239 nM (Sigma-2 receptor)

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Canonical SMILES	CC1=C(C(=NC(=N1)C2=CC=C(C=C2)F)OCCCN3CCCCC3)Cl
Molecular Weight	363.86

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