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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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S335708-1mg | 1mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $55.90 | |
S335708-5mg | 5mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $171.90 | |
S335708-10mg | 10mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $285.90 | |
S335708-25mg | 25mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $589.90 | |
S335708-50mg | 50mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $773.90 |
a potent and selective agonist of the 5-HT6 receptor
Synonyms | ST 1936 | 5-Chloro-3-[2-(dimethylamino)ethyl] -2-methylindole |
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Specifications & Purity | ≥98% |
Storage Temp | Store at -20°C |
Shipped In | Ice chest + Ice pads |
Product Description | ST1936 is a selective, nanomolar affinity 5-HT6 receptor agonist with Ki values of 13 nM, 168 nM and 245 nM for human 5-HT6, 5-HT7 and 5-HT2B receptors, respectively. ST1936 also shows moderate affinity (Ki of 300 nM) for human and rat α2 adrenergic receptor. |
Ki Data | SR-6: Ki= 13 nM (human); SR-7: Ki= 168 nM (human); SR-2B: Ki= 245 nM (human); α2 adrenergic receptors : Ki= 300 nM (human) |
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IUPAC Name | 2-(5-chloro-2-methyl-1H-indol-3-yl)-N,N-dimethylethanamine |
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INCHI | InChI=1S/C13H17ClN2/c1-9-11(6-7-16(2)3)12-8-10(14)4-5-13(12)15-9/h4-5,8,15H,6-7H2,1-3H3 |
InChi Key | KSYMELKKLOFABL-UHFFFAOYSA-N |
Canonical SMILES | CC1=C(C2=C(N1)C=CC(=C2)Cl)CCN(C)C |
Isomeric SMILES | CC1=C(C2=C(N1)C=CC(=C2)Cl)CCN(C)C |
WGK Germany | 3 |
PubChem CID | 9921064 |
Molecular Weight | 236.74 |
Enter Lot Number to search for COA:
To view the certificate results,please click on a Lot number.For Lot numbers from past orders,please use our order status section
Lot Number | Certificate Type | Date | Item |
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D2403529 | Certificate of Analysis | Mar 18, 2024 | S335708 |
D2403543 | Certificate of Analysis | Mar 18, 2024 | S335708 |
D2403544 | Certificate of Analysis | Mar 18, 2024 | S335708 |
D2403545 | Certificate of Analysis | Mar 18, 2024 | S335708 |
D2403546 | Certificate of Analysis | Mar 18, 2024 | S335708 |
D2403547 | Certificate of Analysis | Mar 18, 2024 | S335708 |
D2403548 | Certificate of Analysis | Mar 18, 2024 | S335708 |
Solubility | Soluble in DMSO (100 mM). |
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Refractive Index | n20D~1.61 (Predicted) |
Hazard Statements | H302:Harmful if swallowed |
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WGK Germany | 3 |
RIDADR | NONHforallmodesoftransport |