TAK-683 acetate - 98%, high purity , CAS No.T658894

  • ≥98%
Item Number
T658894
Grouped product items
SKUSizeAvailabilityPrice Qty
T658894-1mg
1mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$350.90
T658894-5mg
5mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$850.90
T658894-10mg
10mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$1,450.90
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Basic Description

Specifications & Purity≥98%
Storage TempProtected from light,Argon charged,Desiccated,Store at -80°C
Shipped InIce chest + Ice pads
Product Description

TAK-683 acetate is a potent full KISS1 receptor (KISS1R) agonist ( IC 50 =170 pM) with improved metabolic stability. TAK-683 acetate is a nonapeptide metastin analog, exhibits agonistic activities to KISS1R with EC 50 values of 0.96 nM and 1.6 nM for huma

Appearance:Solid

In Vitro:TAK-683 acetate exhibits an IC 50 value (95% CI) from receptor binding assays is 150-180 pM and EC 50 value (95% CI) from Ca + mobilization assays is 180 (159–203) pM in rat KISS1R-expressing Chinese hamster ovary (CHO) cells. MCE has not independent

In Vivo:TAK-683 acetate (subcutaneous injection; 0.008, 0.08, 0.8, or 8 μmol/ml/kg; once daily; 7 days) induces an increase in plasma luteinizing hormone and testosterone levels; however, after day 7, plasma hormone levels and genital organ weights are reduced.

Biological Activity:TAK-683 acetate is a potent full KISS1 receptor (KISS1R) agonist ( IC 50 =170 pM) with improved metabolic stability. TAK-683 acetate is a nonapeptide metastin analog, exhibits agonistic activities to KISS1R with EC 50 values of 0.96 nM and 1.6 nM for huma

Names and Identifiers

Molecular Weight 1358.5

Certificates

Certificate of Analysis(COA)

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Chemical and Physical Properties

SolubilityH2O : 5 mg/mL (3.68 mM; Need ultrasonic)

Related Documents

Solution Calculators