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Protein or Target Summary

G protein-coupled receptor kinase 5

Gene ID2869
uniprotP34947
Gene NameGRK5
Ensernbl IDENSP00000376609
FamilyBelongs to the protein kinase superfamily. AGC Ser/Thr protein kinase family. GPRK subfamily.
Sequence
MELENIVANTVLLKAREGGGGKRKGKSKKWKEILKFPHISQCEDLRRTIDRDYCSLCDKQPIGRLLFRQFCETRPGLECYIQFLDSVAEYEVTPDEKLGEKGKEIMTKYLTPKSPVFIAQVGQDLVSQTEEKLLQKPCKELFSACAQSVHEYLRGEPFHEYLDSMFFDRFLQWKWLERQPVTKNTFRQYRVLGKGGFGEVCACQVRATGKMYACKRLEKKRIKKRKGESMALNEKQILEKVNSQFVVNLAYAYETKDALCLVLTIMNGGDLKFHIYNMGNPGFEEERALFYAAEILCGLEDLHRENTVYRDLKPENILLDDYGHIRISDLGLAVKIPEGDLIRGRVGTVGYMAPEVLNNQRYGLSPDYWGLGCLIYEMIEGQSPFRGRKEKVKREEVDRRVLETEEVYSHKFSEEAKSICKMLLTKDAKQRLGCQEEGAAEVKRHPFFRNMNFKRLEAGMLDPPFVPDPRAVYCKDVLDIEQFSTVKGVNLDHTDDDFYSKFSTGSVSIPWQNEMIETECFKELNVFGPNGTLPPDLNRNHPPEPPKKGLLQRLFKRQHQNNSKSSPSSKTSFNHHINSNHVSSNSTGSS
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Gene and Protein Information

SpeciesGene IDGene SymbolGene NameUniprot
HUMAN2869GRK5G protein-coupled receptor kinase 5P34947
MOUSE14773Grk5G protein-coupled receptor kinaseQ3TST4
MOUSE14773Grk5G protein-coupled receptor kinase 5Q8VEB1
RAT59075Grk5G protein-coupled receptor kinaseQ66HL7
RAT59075Grk5G protein-coupled receptor kinase 5Q62833

Protein Classes

PANTHER Classes
protein    /    non-receptor serine/threonine protein kinase    /    G protein-coupled receptor kinase 5
protein    /    protein kinase    /    G protein-coupled receptor kinase 5
protein    /    transferase    /    G protein-coupled receptor kinase 5
protein    /    kinase    /    G protein-coupled receptor kinase 5
DTO Classes
protein    /    Kinase    /    Protein kinase    /    AGC group    /    GRK family    /    GRK subfamily    /    G protein-coupled receptor kinase 5

Associated Recombinant Proteins

NameSpecification and purityExpression systemProtein labelActivityView Details

Associated Antibodies

NameSpecificationsSpecies reactivityspeciesApplicationView Details

Associated Approved Drugs

    Associated Active Ligands

      Associated Diseases

      NameDisease TypeMondoid

      Pathway

      Data SourceNameExplore more targetsExplore in Source