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MTNR1A

DescriptionMelatonin receptor type 1A

Gene and Protein Information

Gene ID4543
Uniprot Accession IDs A0AVC5 B0M0L2 Mel-1A-R
Ensembl ID ENSP00000302811
Symbol MT1 MEL-1A-R
FamilyBelongs to the G-protein coupled receptor 1 family.
Sequence
MQGNGSALPNASQPVLRGDGARPSWLASALACVLIFTIVVDILGNLLVILSVYRNKKLRNAGNIFVVSLAVADLVVAIYPYPLVLMSIFNNGWNLGYLHCQVSGFLMGLSVIGSIFNITGIAINRYCYICHSLKYDKLYSSKNSLCYVLLIWLLTLAAVLPNLRAGTLQYDPRIYSCTFAQSVSSAYTIAVVVFHFLVPMIIVIFCYLRIWILVLQVRQRVKPDRKPKLKPQDFRNFVTMFVVFVLFAICWAPLNFIGLAVASDPASMVPRIPEWLFVASYYMAYFNSCLNAIIYGLLNQNFRKEYRRIIVSLCTARVFFVDSSNDVADRVKWKPSPLMTNNNVVKVDSV
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Homologous gene and protein info.
SpeciesGene IDGene SymbolNameTax IDOther Gene IDSources
Chimp471417MTNR1Amelatonin receptor 1A9598OMA, EggNOG
Macaque702686MTNR1Amelatonin receptor 1A9544Inparanoid, OMA, EggNOG
Mouse17773Mtnr1amelatonin receptor 1A10090MGI:102967Inparanoid, OMA, EggNOG
Rat114211Mtnr1amelatonin receptor 1A10116RGD:620797OMA, EggNOG
Horse100056423MTNR1Amelatonin receptor 1A9796VGNC:20432Inparanoid, OMA, EggNOG
Cow539948MTNR1Amelatonin receptor 1A9913VGNC:31746Inparanoid, OMA, EggNOG
OpossumMTNR1Amelatonin receptor 1A [Source:HGNC Symbol;Acc:HGNC:7463]13616Inparanoid, OMA
Chicken396319MTNR1Amelatonin receptor 1A9031CGNC:49752Inparanoid, OMA
Xenopus100488908mtnr1amelatonin receptor 1A8364XB-GENE-1018462Inparanoid, OMA, EggNOG
Zebrafish30667mtnr1aamelatonin receptor 1A a7955ZDB-GENE-990415-155Inparanoid, OMA

Protein Classes

PANTHER Classes
protein    /    receptor    /    G-protein coupled receptor    /    Melatonin receptor type 1a
DTO Classes
protein    /    G-protein coupled receptor    /    Class A rhodopsin like    /    Melatonin receptor    /    Melatonin receptor type 1a

Associated Recombinant Proteins

NameSpecification and purityExpression systemProtein labelAvailabilityView Details

Associated Antibodies

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NameSpecificationsSpecies reactivityApplicationAvailabilityView Details

Associated Approved Drugs

    Associated Active Ligands

      Associated Diseases

      NameDirect Associated TargetsDisease TypeMondoid

      Bibliography

      1.Ebisawa, T T and 19 more authors. 1999-09-07 Alleic variants of human melatonin 1a receptor: function and prevalence in subjects with circadian rhythm sleep disorders. [PMID:10471411]
      2.Roka, F F and 6 more authors. 1999-11 Tight association of the human Mel(1a)-melatonin receptor and G(i): precoupling and constitutive activity. [PMID:10531408]
      3.Brydon, L L and 9 more authors. 1999-12 Dual signaling of human Mel1a melatonin receptors via G(i2), G(i3), and G(q/11) proteins. [PMID:10598579]
      4.Niles, L P LP, Wang, J J, Shen, L L, Lobb, D K DK and Younglai, E V EV. 1999-10-25 Melatonin receptor mRNA expression in human granulosa cells. [PMID:10612428]
      5.Khan, A U AU and Olson, D L DL. 1975-08 Physical therapy and exercise-induced bronchospasm. [PMID:1144527]
      6.Song, C K CK and Bartness, T J TJ. 2001-08 CNS sympathetic outflow neurons to white fat that express MEL receptors may mediate seasonal adiposity. [PMID:11448873]
      7.Roy, D D, Angelini, N L NL, Fujieda, H H, Brown, G M GM and Belsham, D D DD. 2001-11 Cyclical regulation of GnRH gene expression in GT1-7 GnRH-secreting neurons by melatonin. [PMID:11606436]
      8.Savaskan, Egemen E and 8 more authors. 2002-04 Distribution of melatonin MT1 receptor immunoreactivity in human retina. [PMID:11897804]
      9.Ayoub, Mohammed A MA and 6 more authors. 2002-06-14 Monitoring of ligand-independent dimerization and ligand-induced conformational changes of melatonin receptors in living cells by bioluminescence resonance energy transfer. [PMID:11940583]
      10.Yuan, Lin L, Collins, April R AR, Dai, Jun J, Dubocovich, Margarita L ML and Hill, Steven M SM. 2002-06-28 MT(1) melatonin receptor overexpression enhances the growth suppressive effect of melatonin in human breast cancer cells. [PMID:12088876]