Terguride - ≥98%, high purity , CAS No.37686-84-3, Agonist of 5-HT 1A receptor;Agonist of 5-HT 1B receptor;Agonist of 5-HT 1D receptor;Agonist of 5-HT 2A receptor;Antagonist of 5-HT 2B receptor;Antagonist of 5-HT 2C receptor;Antagonist of α 1A-adrenoceptor;Antagonist of α 2A-adrenoceptor;Antagonist of α 2
Terguride - ≥98%, high purity , CAS No.37686-84-3, Agonist of 5-HT 1A receptor;Agonist of 5-HT 1B receptor;Agonist of 5-HT 1D receptor;Agonist of 5-HT 2A receptor;Antagonist of 5-HT 2B receptor;Antagonist of 5-HT 2C receptor;Antagonist of α 1A-adrenoceptor;Antagonist of α 2A-adrenoceptor;Antagonist of α 2
Partial D2 agonist. Potent, non-competitive and non-selective 5-HT 2 antagonist. Shows antiparkinsonism and antidepressant effects in vivo. Blood-brain barrier permeable. Orally active.
Storage Temp
Room temperature,Desiccated
Shipped In
Normal
Grade
Moligand™
Action Type
AGONIST, ANTAGONIST
Mechanism of action
Agonist of 5-HT 1A receptor;Agonist of 5-HT 1B receptor;Agonist of 5-HT 1D receptor;Agonist of 5-HT 2A receptor;Antagonist of 5-HT 2B receptor;Antagonist of 5-HT 2C receptor;Antagonist of α 1A-adrenoceptor;Antagonist of α 2A-adrenoceptor;Antagonist of α 2
Note
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
Product Description
Store at Room Temperature. Store under desiccating conditions. The product can be stored for up to 12 months.
Associated Targets
C8orf49Tdark Putative uncharacterized protein C8orf49 0 Activities
1.Gocht A et al.. (2018) Effects of different serotonin receptor subtype antagonists on the development of cardiac allograft vasculopathy in murine aortic allografts.. Transpl Immunol, [PMID:29649585]
2.Mann A et al.. (2021) New phosphosite-specific antibodies to unravel the role of GRK phosphorylation in dopamine D2 receptor regulation and signaling.. Sci Rep, 11 (8288). [PMID:33859231]
Solution Calculators
Molarity Calculator
Determine the necessary mass, volume, or concentration for preparing a solution.
Dilution Calculator
Determine the dilution needed to prepare a stock solution.