Tesofensine - ≥98%, high purity , Monoamine transporter inhibitor, CAS No.195875-84-4, Monoamine transporter inhibitor

Item Number

T342495

Grouped product items
SKU	Size	Availability	Price
T342495-1mg	1mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$93.90
T342495-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$290.90
T342495-10mg	10mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$522.90
T342495-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$978.90
T342495-50mg	50mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,369.90

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Basic Description

Synonyms	Tesofensine\|195875-84-4\|NS-2330\|Tesofensine [INN]\|BLH9UKX9V1\|NS 2330\|(1R,2R,3S,5S)-3-(3,4-dichlorophenyl)-2-(ethoxymethyl)-8-methyl-8-azabicyclo[3.2.1]octane\|NS2330\|(1R,2R,3S,5S)-3-(3,4-Dichlorophenyl)-2-(ethoxymethyl)-8-methyl-8-azabicyclo(3.2.1)octane\|U
Specifications & Purity	≥98%
Storage Temp	Store at 2-8°C,Protected from light
Shipped In	Wet ice
Action Type	INHIBITOR
Mechanism of action	Monoamine transporter inhibitor
Product Description	Tesofensine (NS-2330) is a triple monoamine reuptake inhibitor inducing a potent inhibition of the re-uptake process in the synaptic cleft of the neurotransmitters dopamine (DA; IC50=6.5 nM), norepinephrine (NE;IC50=1.7 nM), and serotonin (5-HT;IC50=11 nM), and with potentials as an anti-obesity agent. Tesofensine is a CNS acting anti-obesity agent.

Names and Identifiers

IUPAC Name	(1R,2R,3S,5S)-3-(3,4-dichlorophenyl)-2-(ethoxymethyl)-8-methyl-8-azabicyclo[3.2.1]octane
INCHI	InChI=1S/C17H23Cl2NO/c1-3-21-10-14-13(9-12-5-7-17(14)20(12)2)11-4-6-15(18)16(19)8-11/h4,6,8,12-14,17H,3,5,7,9-10H2,1-2H3/t12-,13+,14+,17+/m0/s1
InChi Key	VCVWXKKWDOJNIT-ZOMKSWQUSA-N
Canonical SMILES	CCOCC1C2CCC(N2C)CC1C3=CC(=C(C=C3)Cl)Cl
Isomeric SMILES	CCOC[C@H]1[C@H]2CC[C@H](N2C)C[C@@H]1C3=CC(=C(C=C3)Cl)Cl
PubChem CID	11370864
Molecular Weight	328.28

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Basic Description