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G protein-coupled receptors (GPCRs)
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TG8-260 - 98%, high purity , CAS No.2490544-50-6, Antagonist of EP 2 receptor

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TG8-260 - 98%, high purity , CAS No.2490544-50-6, Antagonist of EP 2 receptor

Moligand™
≥98%

CAS#: 2490544-50-6
Formula: C₂₁H₂₀N₄O
Molecular Weight: 344.41

Item Number

T614409

Grouped product items
SKU	Size	Availability	Price	Qty
T614409-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$674.90
T614409-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,020.90

View related series

EP2 receptor Antagonist Prostaglandin E2 receptor antagonist

Basic Description

Synonyms	compound 2f;TG8260
Specifications & Purity	98%
Storage Temp	Store at -20°C,Argon charged
Shipped In	Ice chest + Ice pads
Grade	Moligand™
Action Type	ANTAGONIST
Mechanism of action	Antagonist of EP 2 receptor

Associated Targets

PTGER2 Tclin Prostaglandin E2 receptor EP2 subtype 0 Activities

Discover Target: PTGER2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

Molecular Weight	344.41

Database links

PubChem CID	155128767

Certificates

Certificate of Analysis(COA)

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4 results found

Lot Number	Certificate Type	Date	Item
C2425551	Certificate of Analysis	Feb 04, 2024	T614409
C2425552	Certificate of Analysis	Feb 04, 2024	T614409
C2425573	Certificate of Analysis	Feb 04, 2024	T614409
C2425574	Certificate of Analysis	Feb 04, 2024	T614409

References

1. Amaradhi R, Mohammed S, Banik A, Franklin R, Dingledine R, Ganesh T. (2022) Second-Generation Prostaglandin Receptor EP2 Antagonist, TG8-260, with High Potency, Selectivity, Oral Bioavailability, and Anti-Inflammatory Properties.. ACS Pharmacol Transl Sci, 5 (2): (118-133). [PMID:35187419]

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