THZ1-R - 10mM in DMSO, high purity , CAS No.1621523-07-6(DMSO)

Item Number

T654558

• Specifications & Purity: 10mM in DMSO
• Storage Temp: Store at -80°C
• Shipped In: Ice chest + Ice pads

Product Description

THZ1-R is a non-cysteine reactive analog of THZ1 which displays diminished activity for CDK7 inhibition. THZ1-R binds to CDK7 with a K d of 142 nM.

In Vitro

THZ1-R shows lower affinity at CDK7 than THZ1, with IC 50 of 146 nM. MCE has not independently confirmed the accuracy of these methods. They are for reference only.

IC50& Target:CDK7 146 nM (IC 50 )