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G protein-coupled receptors (GPCRs)
Opioid receptors
TRAP-101 , CAS No.T614526, Antagonist of NOP receptor

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TRAP-101 , CAS No.T614526, Antagonist of NOP receptor

Moligand™

PubChem CID: 11494970

Item Number

T614526

Grouped product items
SKU	Size	Availability	Price	Qty
T614526-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$670.90
T614526-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90

View related series

NOP receptor Antagonist

Basic Description

Synonyms	Trap101
Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	ANTAGONIST
Mechanism of action	Antagonist of NOP receptor

Associated Targets

HDAC6 Tclin Histone deacetylase 6 0 Activities

Discover Target: HDAC6

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

OPRL1 Tchem Nociceptin receptor 0 Activities

Discover Target: OPRL1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	1-[1-(cyclooctylmethyl)-5-(hydroxymethyl)-3,6-dihydro-2H-pyridin-4-yl]-3-ethylbenzimidazol-2-one
INCHI	InChI=1S/C24H35N3O2/c1-2-26-22-12-8-9-13-23(22)27(24(26)29)21-14-15-25(17-20(21)18-28)16-19-10-6-4-3-5-7-11-19/h8-9,12-13,19,28H,2-7,10-11,14-18H2,1H3
InChi Key	DCRGHMJXEBSRQG-UHFFFAOYSA-N
Canonical SMILES	OCC1=C(CCN(C1)CC1CCCCCCC1)n1c(=O)n(c2c1cccc2)CC
Isomeric SMILES	CCN1C2=CC=CC=C2N(C1=O)C3=C(CN(CC3)CC4CCCCCCC4)CO
PubChem CID	11494970

Database links

PubChem CID	11494970
ChEMBL Ligand	CHEMBL3182208
GPCRdb Ligand	TRAP-101

Certificates

Certificate of Analysis(COA)

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References

1. Trapella C, Guerrini R, Piccagli L, Calo' G, Carra' G, Spagnolo B, Rubini S, Fanton G, Hebbes C, McDonald J et al.. (2006) Identification of an achiral analogue of J-113397 as potent nociceptin/orphanin FQ receptor antagonist.. Bioorg Med Chem, 14 (3): (692-704). [PMID:16202610]

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