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Tropisetron - 99%, high purity , CAS No.89565-68-4, Antagonist of 5-HT 3A;Antagonist of 5-HT 4 receptor;Antagonist of glycine receptor α1 subunit;Antagonist of glycine receptor α2 subunit;Antagonist of glycine receptor β subunit

Moligand™
≥99%

CAS#: 89565-68-4
Formula: C₁₇H₂₀N₂O₂
Molecular Weight: 284.35
PubChem CID: 656665

Item Number

T127885

Grouped product items
SKU	Size	Availability	Price	Qty
T127885-1g	1g	In stock	$45.90
T127885-5g	5g	In stock	$156.90

View related series

5-HT3A Antagonist 5-HT4 receptor Antagonist Glycine Receptor (All subtypes) Antagonist Glycine Receptor (All subtypes) Subunit-specific glycine receptor α1 subunit Antagonist glycine receptor α2 subunit Antagonist glycine receptor β subunit Antagonist

Basic Description

Synonyms	tropisetron\|89565-68-4\|Navoban\|Tropisetronum\|Novaban\|[(1R,5S)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl] 1H-indole-3-carboxylate\|Tropisteron\|ICS 205930\|Tropisetron (INN)\|(3-endo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl 1H-indole-3-carboxylate\|Navoban (TN)\|ICF 2
Specifications & Purity	99%
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads
Grade	Moligand™
Action Type	ANTAGONIST
Mechanism of action	Antagonist of 5-HT 3A;Antagonist of 5-HT 4 receptor;Antagonist of glycine receptor α1 subunit;Antagonist of glycine receptor α2 subunit;Antagonist of glycine receptor β subunit

Associated Targets

GLRA2 Tchem Glycine receptor subunit alpha-2 1 Activities

Discover Target: GLRA2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

HTR4 Tclin 5-hydroxytryptamine receptor 4 2 Activities

Discover Target: HTR4

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

HTR3A Tclin 5-hydroxytryptamine receptor 3A 4 Activities

Discover Target: HTR3A

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

GLRA1 Tclin Glycine receptor subunit alpha-1 1 Activities

Discover Target: GLRA1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

GLRB Tclin Glycine receptor subunit beta 1 Activities

Discover Target: GLRB

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	[(1R,5S)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl] 1H-indole-3-carboxylate
INCHI	InChI=1S/C17H20N2O2/c1-19-11-6-7-12(19)9-13(8-11)21-17(20)15-10-18-16-5-3-2-4-14(15)16/h2-5,10-13,18H,6-9H2,1H3/t11-,12+,13?
InChi Key	ZNRGQMMCGHDTEI-FUNVUKJBSA-N
Canonical SMILES	CN1C2CCC1CC(C2)OC(=O)C3=CNC4=CC=CC=C43
Isomeric SMILES	CN1[C@@H]2CC[C@H]1CC(C2)OC(=O)C3=CNC4=CC=CC=C43
PubChem CID	656665
Molecular Weight	284.35

PubChem CID

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2 results found

Lot Number	Certificate Type	Date	Item
I2226086	Certificate of Analysis	Jul 08, 2024	T127885
I2226170	Certificate of Analysis	Jul 08, 2024	T127885

Safety and Hazards(GHS)

Pictogram(s)	GHS07
Signal	Warning
Hazard Statements	H315:Causes skin irritation H319:Causes serious eye irritation H335:May cause respiratory irritation H302:Harmful if swallowed
Precautionary Statements	P261:Avoid breathing dust/fume/gas/mist/vapors/spray. P305+P351+P338:IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses if present and easy to do - continue rinsing.

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