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Udenafil - 98%, high purity , Phosphodiesterase 5A inhibitor, CAS No.268203-93-6, Phosphodiesterase 5A inhibitor

Moligand™
≥98%

CAS#: 268203-93-6
Formula: C₂₅H₃₆N₆O₄S
Molecular Weight: 516.66
PubChem CID: 135413547

Item Number

U333275

Grouped product items
SKU	Size	Availability	Price
U333275-50mg	50mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$528.90
U333275-250mg	250mg	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$2,380.90
U333275-1g	1g	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$8,569.90

PDE5A (phosphodiesterase 5) inhibitor.

View related series

phosphodiesterase 5A Inhibitor

Basic Description

Synonyms	Udenafil\|268203-93-6\|Zydena\|DA-8159\|L5IB4XLY36\|3-(1-methyl-7-oxo-3-propyl-4H-pyrazolo[4,3-d]pyrimidin-5-yl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-propoxybenzenesulfonamide\|CID 6918523\|3-(1-methyl-7-oxo-3-propyl-4,7-dihydro-1H-pyrazolo(4,3-d)pyrimidin-5-y
Specifications & Purity	98%
Storage Temp	Store at 2-8°C
Shipped In	Wet ice
Grade	Moligand™
Action Type	INHIBITOR
Mechanism of action	Phosphodiesterase 5A inhibitor
Product Description	Udenafil is an oral phosphodiesterase 5 inhibitor.

pKa

pKₐ: 3.5 (Predicted)

ALogP

Names and Identifiers

IUPAC Name	3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-propoxybenzenesulfonamide
INCHI	InChI=1S/C25H36N6O4S/c1-5-8-20-22-23(31(4)29-20)25(32)28-24(27-22)19-16-18(10-11-21(19)35-15-6-2)36(33,34)26-13-12-17-9-7-14-30(17)3/h10-11,16-17,26H,5-9,12-15H2,1-4H3,(H,27,28,32)
InChi Key	IYFNEFQTYQPVOC-UHFFFAOYSA-N
Canonical SMILES	CCCC1=NN(C2=C1N=C(NC2=O)C3=C(C=CC(=C3)S(=O)(=O)NCCC4CCCN4C)OCCC)C
Isomeric SMILES	CCCC1=NN(C2=C1N=C(NC2=O)C3=C(C=CC(=C3)S(=O)(=O)NCCC4CCCN4C)OCCC)C
PubChem CID	135413547
Molecular Weight	516.66

PubChem CID

CAS Registry No.

ChEMBL Ligand

DrugBank Ligand

Certificates

Certificate of Analysis(COA)

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4 results found

Lot Number	Certificate Type	Date	Item
B2426260	Certificate of Analysis	Jun 20, 2022	U333275
H2224316	Certificate of Analysis	Jun 20, 2022	U333275
H2224361	Certificate of Analysis	Jun 20, 2022	U333275
H2224541	Certificate of Analysis	Jun 20, 2022	U333275

Solubility

Soluble in chloroform, and methanol.

Melt Point(°C)

154.0-155.0° C

References

1. Oh TY, Kang KK, Ahn BO, Yoo M, Kim WB. (2000) Erectogenic effect of the selective phosphodiesterase type 5 inhibitor, DA-8159.. Arch Pharm Res, 23 (5): (471-6). [PMID:11059826]
2. Shim HJ, Lee EJ, Kim SH, Kim SH, Yoo M, Kwon JW, Kim WB, Lee HS, Lee MG. (2000) Pharmacokinetics, stability, and blood partition of DA-8159, a new phosphodiesterase V inhibitor.. Res Commun Mol Pathol Pharmacol, 108 (3-4): (275-86). [PMID:11913718]
3. Ahn BO, Kang KK, Ahn GJ, Kwon JW, Kim WB, Kang KS, Lee YS. (2003) Efficacy of DA-8159, a new PDE5 inhibitor, for inducing penile erection in rabbits with acute spinal cord injury.. Int J Impot Res, 15 (6): (405-11). [PMID:14671658]

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Udenafil - 98%, high purity , Phosphodiesterase 5A inhibitor, CAS No.268203-93-6, Phosphodiesterase 5A inhibitor

Basic Description

Product Properties

Associated Targets

PDE5A Tclin cGMP-specific 3',5'-cyclic phosphodiesterase 0 Activities

Names and Identifiers

Database links

Certificates

Certificate of Analysis(COA)

Chemical and Physical Properties

Related Documents

References

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