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Varenicline - 98% , high purity , Neuronal acetylcholine receptor; alpha4/beta2 partial agonist, CAS No.249296-44-4, Neuronal acetylcholine receptor; alpha4/beta2 partial agonist

Moligand™
≥98%

CAS#: 249296-44-4
Formula: C₁₃H₁₃N₃
Molecular Weight: 211.26
PubChem CID: 170361

Item Number

V125892

Grouped product items
SKU	Size	Availability	Price
V125892-5mg	5mg	In stock	$82.90
V125892-10mg	10mg	In stock	$117.90
V125892-25mg	25mg	In stock	$224.90
V125892-50mg	50mg	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$355.90
V125892-100mg	100mg	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$593.90

View related series

nicotinic acetylcholine receptor α3 subunit Agonist nicotinic acetylcholine receptor α4 subunit Agonist

Basic Description

Synonyms	Varenicline\|249296-44-4\|6,10-Methano-6H-pyrazino[2,3-h][3]benzazepine, 7,8,9,10-tetrahydro-\|5,8,14-triazatetracyclo[10.3.1.02,11.04,9]hexadeca-2,4,6,8,10-pentaene\|Varenicline (INN)\|CHEMBL556954\|CP-526555\|NCGC00247735-01\|NCGC00247735-02\|CHEMBL1396\|SCHEMBL2
Specifications & Purity	98%
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads
Grade	Moligand™
Action Type	AGONIST, PARTIAL AGONIST
Mechanism of action	Neuronal acetylcholine receptor; alpha4/beta2 partial agonist

Associated Targets

CHRNA7 Tchem Neuronal acetylcholine receptor subunit alpha-7 1 Activities

Discover Target: CHRNA7

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

CHRNA3 Tclin Neuronal acetylcholine receptor subunit alpha-3 0 Activities

Discover Target: CHRNA3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

CHRNA4 Tclin Neuronal acetylcholine receptor subunit alpha-4 1 Activities

Discover Target: CHRNA4

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	5,8,14-triazatetracyclo[10.3.1.02,11.04,9]hexadeca-2,4,6,8,10-pentaene
INCHI	InChI=1S/C13H13N3/c1-2-16-13-5-11-9-3-8(6-14-7-9)10(11)4-12(13)15-1/h1-2,4-5,8-9,14H,3,6-7H2
InChi Key	JQSHBVHOMNKWFT-UHFFFAOYSA-N
Canonical SMILES	C1C2CNCC1C3=CC4=NC=CN=C4C=C23
Isomeric SMILES	C1C2CNCC1C3=CC4=NC=CN=C4C=C23
PubChem CID	170361
Molecular Weight	211.26

Wikipedia

DrugBank Ligand

CAS Registry No.

PubChem CID

ChEMBL Ligand

ChEBI

RCSB PDB Ligand

PEP

DrugCentral Ligand

Certificates

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5 results found

Lot Number	Certificate Type	Date	Item
C2210175	Certificate of Analysis	Dec 22, 2023	V125892
C2210181	Certificate of Analysis	Dec 22, 2023	V125892
C2210613	Certificate of Analysis	Dec 22, 2023	V125892
C2210636	Certificate of Analysis	Dec 22, 2023	V125892
C2210668	Certificate of Analysis	Dec 22, 2023	V125892

Safety and Hazards(GHS)

Pictogram(s)	GHS09, GHS07
Signal	Warning
Hazard Statements	H302:Harmful if swallowed H400:Very toxic to aquatic life H410:Very toxic to aquatic life with long lasting effects
Precautionary Statements	P273:Avoid release to the environment. P501:Dispose of contents/container to ... P264:Wash hands [and …] thoroughly after handling. P270:Do not eat, drink or smoke when using this product. P391:Collect spillage. P330:Rinse mouth. P301+P317:IF SWALLOWED: Get medical help.

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