Determine the necessary mass, volume, or concentration for preparing a solution.
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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B303612-1g | 1g | In stock | $145.90 | |
B303612-5g | 5g | In stock | $654.90 | |
B303612-25g | 25g | In stock | $2,943.90 |
Synonyms | 1-Butyl-2',6'-pipecoloxylidide | AH250 | AH-250 | BPBio1_000298 | Exparel (TN) | KBio2_007140 | LAC-43 | SCHEMBL25438 | AKOS016842516 | EINECS 218-553-3 | Liposomal bupivacaine | Bupivacaine liposome | Spectrum3_000974 | 1-butyl-N-(2,6-dimethylphenyl)-pip |
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Specifications & Purity | Moligand™, ≥97% |
Storage Temp | Store at 2-8°C |
Shipped In | Wet ice |
Grade | Moligand™ |
Action Type | CHANNEL BLOCKER, GATING INHIBITOR |
Mechanism of action | Gating inhibitor of K ir3.2;Channel blocker of K v1.5;Channel blocker of K v4.3;Channel blocker of Na v1.5 |
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Mechanism of Action | Action Type | target ID | Target Name | Target Type | Target Organism | Binding Site Name | References |
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Glucocorticoid receptor agonist | AGONIST | ALA2034 | Glucocorticoid receptor | SINGLE PROTEIN | Homo sapiens | ||
Glucocorticoid receptor agonist | AGONIST | ALA2034 | Glucocorticoid receptor | SINGLE PROTEIN | Homo sapiens | ||
Glucocorticoid receptor agonist | AGONIST | ALA2034 | Glucocorticoid receptor | SINGLE PROTEIN | Homo sapiens | PubMed: [1] | |
Glucocorticoid receptor agonist | AGONIST | ALA2034 | Glucocorticoid receptor | SINGLE PROTEIN | Homo sapiens | PubMed: [1] | |
Glucocorticoid receptor agonist | AGONIST | ALA2034 | Glucocorticoid receptor | SINGLE PROTEIN | Homo sapiens | ||
Glucocorticoid receptor agonist | AGONIST | ALA2034 | Glucocorticoid receptor | SINGLE PROTEIN | Homo sapiens | ||
Glucocorticoid receptor agonist | AGONIST | ALA2034 | Glucocorticoid receptor | SINGLE PROTEIN | Homo sapiens | ||
Glucocorticoid receptor agonist | AGONIST | ALA2034 | Glucocorticoid receptor | SINGLE PROTEIN | Homo sapiens | ||
Glucocorticoid receptor agonist | AGONIST | ALA2034 | Glucocorticoid receptor | SINGLE PROTEIN | Homo sapiens | PubMed: [1] | |
Glucocorticoid receptor agonist | AGONIST | ALA2034 | Glucocorticoid receptor | SINGLE PROTEIN | Homo sapiens |
IUPAC Name | 1-butyl-N-(2,6-dimethylphenyl)piperidine-2-carboxamide |
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INCHI | InChI=1S/C18H28N2O/c1-4-5-12-20-13-7-6-11-16(20)18(21)19-17-14(2)9-8-10-15(17)3/h8-10,16H,4-7,11-13H2,1-3H3,(H,19,21) |
InChi Key | LEBVLXFERQHONN-UHFFFAOYSA-N |
Canonical SMILES | CCCCN1CCCCC1C(=O)NC2=C(C=CC=C2C)C |
Isomeric SMILES | CCCCN1CCCCC1C(=O)NC2=C(C=CC=C2C)C |
PubChem CID | 2474 |
Molecular Weight | 288.43 |
PubChem CID | 2474 |
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ChEBI | CHEBI:3215 |
CAS Registry No. | 38396-39-3 |
Wikipedia | Bupivacaine |
ChEMBL Ligand | CHEMBL1098 |
DrugBank Ligand | DB00297 |
BindingDB Ligand | 50017664 |
PEP | bupivacaine |
DrugCentral Ligand | 432 |
Enter Lot Number to search for COA:
Find and download the COA for your product by matching the lot number on the packaging.
4 results found
Lot Number | Certificate Type | Date | Item |
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A2219286 | Certificate of Analysis | Nov 19, 2024 | B303612 |
A2219394 | Certificate of Analysis | Nov 19, 2024 | B303612 |
A2219396 | Certificate of Analysis | Nov 19, 2024 | B303612 |
A2425121 | Certificate of Analysis | Jan 04, 2022 | B303612 |
Solubility | DMSO (Slightly), Methanol (Slightly) |
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Melt Point(°C) | >103ºC |
Pictogram(s) | GHS06 |
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Signal | Danger |
Hazard Statements | H300:Fatal if swallowed H310:Fatal in contact with skin H330:Fatal if inhaled |
Precautionary Statements | P280:Wear protective gloves/protective clothing/eye protection/face protection. P302+P352:IF ON SKIN: wash with plenty of water. P321:Specific treatment (see ... on this label). P405:Store locked up. P501:Dispose of contents/container to ... P264:Wash hands [and …] thoroughly after handling. P260:Do not breathe dust/fume/gas/mist/vapors/spray. P284:[In case of inadequate ventilation] Wear respiratory protection. P271:Use only outdoors or in a well-ventilated area. P270:Do not eat, drink or smoke when using this product. P304+P340:IF INHALED: Remove person to fresh air and keep comfortable for breathing. P403+P233:Store in a well-ventilated place. Keep container tightly closed. P330:Rinse mouth. P262:Do not get in eyes, on skin, or on clothing. P320:Specific treatment is urgent (see ... on this label). P361+P364:Take off immediately all contaminated clothing and wash it before reuse. P301+P316:IF SWALLOWED: Get emergency medical help immediately. P316:Get emergency medical help immediately. |
1. Ying Deng, Jing-Shu Hong, Yi-Yun Cao, Ning Kang, Deng-Yang Han, Yi-Tong Li, Lei Chen, Zheng-Qian Li, Rui Zhan, Xiang-Yang Guo, Ning Yang, Cheng-Mei Shi. (2023) Specific antagonist of receptor for advanced glycation end‑products attenuates delirium‑like behaviours induced by sevoflurane anaesthesia with surgery in aged mice partially by improving damage to the blood‑brain barrier. Experimental and Therapeutic Medicine, 26 (1): (1-10). [PMID:] [10.3892/etm.2023.12016] |
1. Ying Deng, Jing-Shu Hong, Yi-Yun Cao, Ning Kang, Deng-Yang Han, Yi-Tong Li, Lei Chen, Zheng-Qian Li, Rui Zhan, Xiang-Yang Guo, Ning Yang, Cheng-Mei Shi. (2023) Specific antagonist of receptor for advanced glycation end‑products attenuates delirium‑like behaviours induced by sevoflurane anaesthesia with surgery in aged mice partially by improving damage to the blood‑brain barrier. Experimental and Therapeutic Medicine, 26 (1): (1-10). [PMID:] [10.3892/etm.2023.12016] |