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3-(1,2,3-benzothiadiazol-6-yl)-1-[2-(cyclohex-1-en-1-yl)ethyl]urea , CAS No.B608883, Inhibitor of protein arginine methyltransferase 3

3-(1,2,3-benzothiadiazol-6-yl)-1-[2-(cyclohex-1-en-1-yl)ethyl]urea , CAS No.B608883, Inhibitor of protein arginine methyltransferase 3

Item Number

B608883

Grouped product items
SKU	Size	Availability	Price	Qty
B608883-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$700.90
B608883-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90

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Basic Description

Synonyms	compound 1 (allosteric);compound 1
Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	INHIBITOR
Mechanism of action	Inhibitor of protein arginine methyltransferase 3

PRMT3 Tchem Protein arginine N-methyltransferase 3 (1 Activities)

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

PRMT3 Tchem Protein arginine N-methyltransferase 3 (219 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

IUPAC Name	3-(1,2,3-benzothiadiazol-6-yl)-1-[2-(cyclohex-1-en-1-yl)ethyl]urea
INCHI	InChI=1S/C15H18N4OS/c20-15(16-9-8-11-4-2-1-3-5-11)17-12-6-7-13-14(10-12)21-19-18-13/h4,6-7,10H,1-3,5,8-9H2,(H2,16,17,20)
InChi Key	GGXCUZHEJUJACD-UHFFFAOYSA-N
Canonical SMILES	O=C(Nc1ccc2c(c1)snn2)NCCC1=CCCCC1
Isomeric SMILES	C1CCC(=CC1)CCNC(=O)NC2=CC3=C(C=C2)N=NS3
PubChem CID	53346504

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1. Siarheyeva A, Senisterra G, Allali-Hassani A, Dong A, Dobrovetsky E, Wasney GA, Chau I, Marcellus R, Hajian T, Liu F et al.. (2012) An allosteric inhibitor of protein arginine methyltransferase 3.. Structure, 20 (8): (1425-35). [PMID:22795084]

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