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(6E)-6-[(2E)-2-(1H-quinolin-2-ylidene)ethylidene]cyclohexa-2,4-dien-1-one , CAS No.E608873, Inhibitor of Endothelin-converting enzyme 2

(6E)-6-[(2E)-2-(1H-quinolin-2-ylidene)ethylidene]cyclohexa-2,4-dien-1-one , CAS No.E608873, Inhibitor of Endothelin-converting enzyme 2

Item Number

E608873

Grouped product items
SKU	Size	Availability	Price	Qty
E608873-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$600.90
E608873-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90

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Basic Description

Synonyms	compound 1
Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	INHIBITOR
Mechanism of action	Inhibitor of Endothelin-converting enzyme 2

ECE2 Tchem Endothelin-converting enzyme 2 (1 Activities)

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

ECE2 Tchem Endothelin-converting enzyme 2 (7 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

IUPAC Name	(6E)-6-[(2E)-2-(1H-quinolin-2-ylidene)ethylidene]cyclohexa-2,4-dien-1-one
INCHI	InChI=1S/C17H13NO/c19-17-8-4-2-6-14(17)10-12-15-11-9-13-5-1-3-7-16(13)18-15/h1-12,19H/b12-10-
InChi Key	NXNDEWNGCMCWMA-BENRWUELSA-N
Canonical SMILES	Oc1ccccc1/C=C\c1ccc2c(n1)cccc2
Isomeric SMILES	C1=CC=C2C(=C1)C=CC(=N2)/C=C\C3=CC=CC=C3O
PubChem CID	136045796

ChEMBL Ligand	CHEMBL487942
PubChem CID	136045796

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1. Gagnidze K, Sachchidanand, Rozenfeld R, Mezei M, Zhou MM, Devi LA. (2008) Homology modeling and site-directed mutagenesis to identify selective inhibitors of endothelin-converting enzyme-2.. J Med Chem, 51 (12): (3378-87). [PMID:18507370]

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