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Applications
Targets
G protein-coupled receptors (GPCRs)
Bombesin receptors
AM-37 , CAS No.A607583, Antagonist of BB 2 receptor

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AM-37 , CAS No.A607583, Antagonist of BB 2 receptor

Moligand™

PubChem CID: 122181321

Item Number

A607583

Grouped product items
SKU	Size	Availability	Price	Qty
A607583-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,334.90
A607583-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90

View related series

BB2 receptor Antagonist

Basic Description

Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	ANTAGONIST
Mechanism of action	Antagonist of BB 2 receptor

Associated Targets

FPR1 Tchem fMet-Leu-Phe receptor 0 Activities

Discover Target: FPR1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

FPR2 Tchem N-formyl peptide receptor 2 0 Activities

Discover Target: FPR2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

GRPR Tchem Gastrin-releasing peptide receptor 0 Activities

Discover Target: GRPR

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	(2R)-3-(1H-indol-3-yl)-2-[(4-methoxyphenyl)carbamoylamino]-N-[(1-pyridin-3-ylcyclohexyl)methyl]propanamide
INCHI	InChI=1S/C31H35N5O3/c1-39-25-13-11-24(12-14-25)35-30(38)36-28(18-22-19-33-27-10-4-3-9-26(22)27)29(37)34-21-31(15-5-2-6-16-31)23-8-7-17-32-20-23/h3-4,7-14,17,19-20,28,33H,2,5-6,15-16,18,21H2,1H3,(H,34,37)(H2,35,36,38)/t28-/m1/s1
InChi Key	INNVRNIOVHJSQS-MUUNZHRXSA-N
Canonical SMILES	COc1ccc(cc1)NC(=O)N[C@@H](C(=O)NCC1(CCCCC1)c1cccnc1)Cc1c[nH]c2c1cccc2
Isomeric SMILES	COC1=CC=C(C=C1)NC(=O)N[C@H](CC2=CNC3=CC=CC=C32)C(=O)NCC4(CCCCC4)C5=CN=CC=C5
PubChem CID	122181321

Database links

PubChem CID	122181321
BindingDB Ligand	50097560
ChEMBL Ligand	CHEMBL3590072
GPCRdb Ligand	AM-37

Certificates

Certificate of Analysis(COA)

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References

1. Moody TW, Tashakkori N, Mantey SA, Moreno P, Ramos-Alvarez I, Leopoldo M, Jensen RT. (2017) AM-37 and ST-36 Are Small Molecule Bombesin Receptor Antagonists.. Front Endocrinol (Lausanne), 8 (3): (176). [PMID:28785244]

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