Basic Description

Specifications & Purity	96%
Storage Temp	Store at 2-8°C,Protected from light
Shipped In	Wet ice
Product Description	AP-III-a4 (ENOblock) is the first nonsubstrate analogue inhibitor of enolase with IC50 of 0.576 μM.

Associated Targets(Human)

ENO1 Tchem Alpha-enolase (1 Activities)

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

ENO1 Tchem Alpha enolase (27 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

rep Replicase polyprotein 1ab (378 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

SARS-CoV-2 (38078 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

IUPAC Name	N-[2-[2-(2-aminoethoxy)ethoxy]ethyl]-2-[4-[[4-(cyclohexylmethylamino)-6-[(4-fluorophenyl)methylamino]-1,3,5-triazin-2-yl]amino]phenyl]acetamide
INCHI	InChI=1S/C31H43FN8O3/c32-26-10-6-25(7-11-26)22-36-30-38-29(35-21-24-4-2-1-3-5-24)39-31(40-30)37-27-12-8-23(9-13-27)20-28(41)34-15-17-43-19-18-42-16-14-33/h6-13,24H,1-5,14-22,33H2,(H,34,41)(H3,35,36,37,38,39,40)
InChi Key	MOVYITHKOHMLHC-UHFFFAOYSA-N
Canonical SMILES	C1CCC(CC1)CNC2=NC(=NC(=N2)NCC3=CC=C(C=C3)F)NC4=CC=C(C=C4)CC(=O)NCCOCCOCCN
Isomeric SMILES	C1CCC(CC1)CNC2=NC(=NC(=N2)NCC3=CC=C(C=C3)F)NC4=CC=C(C=C4)CC(=O)NCCOCCOCCN
PubChem CID	24012277
Molecular Weight	594.72

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3 results found

Lot Number	Certificate Type	Date	Item
K2223124	Certificate of Analysis	Jul 27, 2022	A418547
K2223154	Certificate of Analysis	Jul 27, 2022	A418547
K2223168	Certificate of Analysis	Jul 27, 2022	A418547

Solubility	DMSO : 62.5 mg/mL (105.09 mM; ultrasonic and warming and heat to 60°C)
Sensitivity	Light sensitive

Signal	Warning
Hazard Statements	H315:Causes skin irritation H319:Causes serious eye irritation H335:May cause respiratory irritation H302:Harmful if swallowed
Precautionary Statements	P261:Avoid breathing dust/fume/gas/mist/vapors/spray. P305+P351+P338:IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses if present and easy to do - continue rinsing.

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SKU	Size	Availability	Price
A418547-5mg	5mg	In stock	$206.90
A418547-25mg	25mg	In stock	$672.90
A418547-100mg	100mg	In stock	$2,422.90