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ARI-3099 , CAS No.A607725, Inhibitor of acylaminoacyl-peptide hydrolase;Inhibitor of fibroblast activation protein alpha

Item Number
A607725
Grouped product items
SKUSizeAvailabilityPrice Qty
A607725-5mg
5mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$1,334.90
A607725-25mg
25mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$2,000.90
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acylaminoacyl-peptide hydrolase Inhibitor fibroblast activation protein alpha Inhibitor

Basic Description

Synonymscompound 226;compound 6;Py(D)AlaboroPro
Specifications & PurityMoligand™
GradeMoligand™
Action TypeINHIBITOR
Mechanism of actionInhibitor of acylaminoacyl-peptide hydrolase;Inhibitor of fibroblast activation protein alpha

Associated Targets(Human)

FAP Tchem Prolyl endopeptidase FAP (4 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)
APEH Tchem Acylamino-acid-releasing enzyme (1 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)
PREP Tchem Prolyl endopeptidase (2 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)
DPP7 Tchem Dipeptidyl peptidase II (2000 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
DPP8 Tchem Dipeptidyl peptidase VIII (2139 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
DPP9 Tchem Dipeptidyl peptidase IX (1624 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
HEK293 (82097 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
FAP Tchem Fibroblast activation protein alpha (827 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID

Associated Targets(non-human)

DPP4 Dipeptidyl peptidase IV (11 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
PREP Prolyl endopeptidase (14 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID

Mechanisms of Action

Mechanism of ActionAction Typetarget IDTarget NameTarget TypeTarget OrganismBinding Site NameReferences

Names and Identifiers

INCHI InChI=1S/C13H18BN3O4/c1-9(16-12(18)10-4-6-15-7-5-10)13(19)17-8-2-3-11(17)14(20)21/h4-7,9,11,20-21H,2-3,8H2,1H3,(H,16,18)/t9-,11+/m1/s1
InChi Key DRBWRJPFNOBNIO-KOLCDFICSA-N
Canonical SMILES OB([C@@H]1CCCN1C(=O)[C@H](NC(=O)c1ccncc1)C)O
Isomeric SMILES B([C@@H]1CCCN1C(=O)[C@@H](C)NC(=O)C2=CC=NC=C2)(O)O
PubChem CID 71655266

Certificates

Certificate of Analysis(COA)

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Related Documents

 SDS

 Specification Sheet

References

1. Poplawski SE, Lai JH, Li Y, Jin Z, Liu Y, Wu W, Wu Y, Zhou Y, Sudmeier JL, Sanford DG et al..  (2013)  Identification of selective and potent inhibitors of fibroblast activation protein and prolyl oligopeptidase..  J Med Chem,  56  (9): (3467-77).  [PMID:23594271] [10.1021/op500134e]
2. Bachovchin DA, Koblan LW, Wu W, Liu Y, Li Y, Zhao P, Woznica I, Shu Y, Lai JH, Poplawski SE et al..  (2014)  A high-throughput, multiplexed assay for superfamily-wide profiling of enzyme activity..  Nat Chem Biol,  10  (8): (656-63).  [PMID:24997602] [10.1021/op500134e]

Solution Calculators

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