Determine the necessary mass, volume, or concentration for preparing a solution.
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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A288879-5mg | 5mg | Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience! | $81.90 | |
A288879-10mg | 10mg | Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience! | $140.90 | |
A288879-25mg | 25mg | Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience! | $271.90 | |
A288879-50mg | 50mg | Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience! | $434.90 | |
A288879-100mg | 100mg | Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience! | $652.90 | |
A288879-250mg | 250mg | Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience! | $1,469.90 | |
A288879-1g | 1g | Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience! | $5,289.90 |
GPR119 receptor agonist
Synonyms | HY-107535 | 2-(2-(4-bromophenyl)-6-methylpyrimidin-4-ylamino)ethanol | DTXSID90416373 | 2-[[2-(4-Bromophenyl)-6-methyl-4-pyrinidinyl]amino]ethanol | 2-[[2-(4-bromophenyl)-6-methylpyrimidin-4-yl]amino]ethanol | AKOS005229115 | Z1095349900 | CS-0028832 | Q2 |
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Specifications & Purity | Moligand™, ≥98%(HPLC) |
Biochemical and Physiological Mechanisms | GPR119 receptor agonist (EC50= 2.5μM in HEK293 cells expressing human GPR119). Enhances insulin secretion stimulated by glucosein vivo. Stimulates proGlukagon gene promoter actvity. Orally available. |
Storage Temp | Protected from light,Store at -20°C |
Shipped In | Ice chest + Ice pads |
Grade | Moligand™ |
Action Type | AGONIST |
Mechanism of action | Agonist of GPR119 |
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Mechanism of Action | Action Type | target ID | Target Name | Target Type | Target Organism | Binding Site Name | References |
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IUPAC Name | 2-[[2-(4-bromophenyl)-6-methylpyrimidin-4-yl]amino]ethanol |
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INCHI | InChI=1S/C13H14BrN3O/c1-9-8-12(15-6-7-18)17-13(16-9)10-2-4-11(14)5-3-10/h2-5,8,18H,6-7H2,1H3,(H,15,16,17) |
InChi Key | DUKPGOOUJNUIOI-UHFFFAOYSA-N |
Canonical SMILES | CC1=CC(=NC(=N1)C2=CC=C(C=C2)Br)NCCO |
Isomeric SMILES | CC1=CC(=NC(=N1)C2=CC=C(C=C2)Br)NCCO |
PubChem CID | 5332859 |
Molecular Weight | 308.17 |
CAS Registry No. | 330981-72-1 |
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PubChem CID | 5332859 |
ChEMBL Ligand | CHEMBL1956589 |
GPCRdb Ligand | AS1269574 |
Enter Lot Number to search for COA:
Find and download the COA for your product by matching the lot number on the packaging.
Lot Number | Certificate Type | Date | Item |
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D2230104 | Certificate of Analysis | Mar 07, 2022 | A288879 |
D2230116 | Certificate of Analysis | Mar 07, 2022 | A288879 |
D2230124 | Certificate of Analysis | Mar 07, 2022 | A288879 |
D2230129 | Certificate of Analysis | Mar 07, 2022 | A288879 |
D2230134 | Certificate of Analysis | Mar 07, 2022 | A288879 |
D2230136 | Certificate of Analysis | Mar 07, 2022 | A288879 |
D2230139 | Certificate of Analysis | Mar 07, 2022 | A288879 |
Solubility | Solvent:DMSO, Max Conc. mg/mL: 30.82, Max Conc. mM: 100; Solvent:ethanol, Max Conc. mg/mL: 30.82, Max Conc. mM: 100 |
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Sensitivity | light sensitive |