astemizole - ≥98%, high purity , Histamine H1 receptor antagonist, CAS No.68844-77-9, Histamine H1 receptor antagonist

Item Number

A133983

• Synonyms: ASTEMIZOLE [USP IMPURITY] | Astemizole,(S) | Retolen | Waruzol | ASTEMIZOLE [VANDF] | Benzimidazole, 1-(p-fluorobenzyl)-2-((1-(2-(p-methoxyphenyl)ethyl)piperid-4-yl)amino)- | ASTEMIZOLE [MART.] | HMS1922L12 | 1-[(4-Fluorophenyl)methyl]-N-{1-[2-(4-methoxyp
• Specifications & Purity: Moligand™, ≥98%
• Biochemical and Physiological Mechanisms: Astermizole is a potent hERG potassium channel blocker (IC50 of 0.9 nM) and may used as a pharmacological chaperone to correct folding defects and restore protein function for some mutated forms of hERG channels. It has also been studied for treatment of
• Storage Temp: Store at 2-8°C,Protected from light
• Shipped In: Wet ice
• Grade: Moligand™
• Action Type: ANTAGONIST, CHANNEL BLOCKER
• Mechanism of action: Histamine H1 receptor antagonist
• Note: Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.