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BIM 23056 - 98%, high purity , CAS No.150155-61-6, Agonist of SST 2 receptor;Agonist of SST 3 receptor;Agonist of SST 5 receptor;Antagonist of SST 5 receptor

Item Number
B275021
Grouped product items
SKUSizeAvailabilityPrice Qty
B275021-1mg
1mg
In stock
$219.90
B275021-5mg
5mg
Available within 4-8 weeks(?)
Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!
$1,111.90
B275021-25mg
25mg
Available within 4-8 weeks(?)
Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!
$5,001.90
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Potent, selective somatostatin receptor 5 (sst 5 ) antagonist

View related series
GPCR/G Protein Neuronal Signaling Somatostatin Receptor SST2 receptor Agonist SST3 receptor Agonist SST5 receptor Agonist SST5 receptor Antagonist

Basic Description

Specifications & PurityMoligand™, ≥98%
Biochemical and Physiological MechanismsPotent, selective somatostatin receptor 5 (sst 5 ) antagonist (K i values are 5.7 (sst 5 ), 10.8 (sst 3 ), 16.6 (sst 4 ), 142 (sst 1 ) and >1000 nM (sst 2 ) for human cloned receptors).
Storage TempStore at -20°C,Desiccated
Shipped InIce chest + Ice pads
GradeMoligand™
Action TypeAGONIST, ANTAGONIST
Mechanism of actionAgonist of SST 2 receptor;Agonist of SST 3 receptor;Agonist of SST 5 receptor;Antagonist of SST 5 receptor
NoteWherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one week. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
Product Description

Store at -20°C. Store under desiccating conditions. The product can be stored for up to 12 months.

Associated Targets(Human)

SSTR2 Tclin Somatostatin receptor type 2 (0 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)
SSTR3 Tclin Somatostatin receptor type 3 (0 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)
SSTR5 Tclin Somatostatin receptor type 5 (0 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

Mechanisms of Action

Mechanism of ActionAction Typetarget IDTarget NameTarget TypeTarget OrganismBinding Site NameReferences

Names and Identifiers

IUPAC Name (2S)-6-amino-N-[(2S)-1-[[(2S)-1-[[(2R)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-amino-3-phenylpropanoyl]amino]-3-phenylpropanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]hexanamide
INCHI InChI=1S/C71H81N11O9/c1-44(2)63(71(91)81-61(39-47-22-10-5-11-23-47)67(87)77-58(64(74)84)41-49-29-32-50-24-12-13-25-51(50)36-49)82-66(86)57(28-16-17-35-72)76-70(90)62(42-52-43-75-56-27-15-14-26-54(52)56)80-69(89)60(40-48-30-33-53(83)34-31-48)79-68(88)59(38-46-20-8-4-9-21-46)78-65(85)55(73)37-45-18-6-3-7-19-45/h3-15,18-27,29-34,36,43-44,55,57-63,75,83H,16-17,28,35,37-42,72-73H2,1-2H3,(H2,74,84)(H,76,90)(H,77,87)(H,78,85)(H,79,88)(H,80,89)(H,81,91)(H,82,86)/t55-,57+,58-,59+,60+,61+,62-,63+/m1/s1
InChi Key VPTPBEUWKCLZGU-OOSWLFMASA-N
Canonical SMILES CC(C)C(C(=O)NC(CC1=CC=CC=C1)C(=O)NC(CC2=CC3=CC=CC=C3C=C2)C(=O)N)NC(=O)C(CCCCN)NC(=O)C(CC4=CNC5=CC=CC=C54)NC(=O)C(CC6=CC=C(C=C6)O)NC(=O)C(CC7=CC=CC=C7)NC(=O)C(CC8=CC=CC=C8)N
Isomeric SMILES CC(C)[C@@H](C(=O)N[C@@H](CC1=CC=CC=C1)C(=O)N[C@H](CC2=CC3=CC=CC=C3C=C2)C(=O)N)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CC4=CNC5=CC=CC=C54)NC(=O)[C@H](CC6=CC=C(C=C6)O)NC(=O)[C@H](CC7=CC=CC=C7)NC(=O)[C@@H](CC8=CC=CC=C8)N
PubChem CID 16133799
Molecular Weight 1232.49

Certificates

Certificate of Analysis(COA)

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4 results found

Lot NumberCertificate TypeDateItem
K2328362Certificate of AnalysisSep 19, 2024 B275021
K2328393Certificate of AnalysisSep 19, 2024 B275021
K2328394Certificate of AnalysisSep 19, 2024 B275021
K2328395Certificate of AnalysisSep 19, 2024 B275021

Chemical and Physical Properties

SolubilitySoluble in 1:2 acetonitrile/water to 20 mg/ml
SensitivityMoisture sensitive

Related Documents

 SDS

 Specification Sheet

Solution Calculators

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