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BX 430 - 10mM in DMSO, high purity , CAS No.688309-70-8
Selective P2X4allosteric antagonist
Basic Description Synonyms N-[2,6-Dibromo-4-(1-methylethyl)phenyl]-N'-(3-pyridinyl)urea；BX430 Specifications & Purity Moligand™, 10mM in DMSO Biochemical and Physiological Mechanisms Selective P2X4allosteric antagonist (IC50= 0.54μM). Exhibits >10-fold selectivity for human P2X4receptors over P2X1, P2X2, P2X3, P2X5and P2X7receptors. Binds noncompetitively at extracellular allosteric site. Effective at human and zebrafish, but not mou Storage Temp Protected from light,Store at -80°C Shipped In Ice chest + Ice pads Grade Moligand™
Associated Targets(Human) Associated Targets(non-human) Names and Identifiers IUPAC Name 1-(2,6-dibromo-4-propan-2-ylphenyl)-3-pyridin-3-ylurea INCHI InChI=1S/C15H15Br2N3O/c1-9(2)10-6-12(16)14(13(17)7-10)20-15(21)19-11-4-3-5-18-8-11/h3-9H,1-2H3,(H2,19,20,21) InChi Key JFNKIJKRXKPQCC-UHFFFAOYSA-N Canonical SMILES CC(C)C1=CC(=C(C(=C1)Br)NC(=O)NC2=CN=CC=C2)Br Isomeric SMILES CC(C)C1=CC(=C(C(=C1)Br)NC(=O)NC2=CN=CC=C2)Br PubChem CID 2810999 Molecular Weight 413.11
Chemical and Physical Properties Sensitivity light sensitive Melt Point(°C) 164-168°C
Safety and Hazards(GHS) RIDADR NONHforallmodesoftransport
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