Calcium-Sensing Receptor Antagonists I - 98%, high purity , CAS No.478963-79-0

  • ≥98%
Item Number
C648197
Grouped product items
SKUSizeAvailabilityPrice Qty
C648197-10mg
10mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$200.90
C648197-50mg
50mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$550.90
C648197-100mg
100mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$850.90
View related series
CaSR GPCR/G Protein

Basic Description

Specifications & Purity≥98%
Biochemical and Physiological MechanismsCalcium-Sensing Receptor Antagonists I is an antagonist of calcium-sensing parathyroid hormone receptors. \nIC50 value:\nTarget: CaSR Calcium-Sensing Receptor Antagonists I is useful for osteoporosis and other bone conditions
Storage TempStore at -20°C
Shipped InIce chest + Ice pads
Product Description

Calcium-Sensing Receptor Antagonists I is an antagonist of calcium-sensing parathyroid hormone receptors.IC50 value:Target: CaSR Calcium-Sensing Receptor Antagonists I is useful for osteoporosis and other bone conditions

Form:Solid

Associated Targets(Human)

CASR Tclin Extracellular calcium-sensing receptor (1 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)
CASR Tclin Calcium sensing receptor (766 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID

Associated Targets(non-human)

Canis familiaris (36305 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
Rattus norvegicus (775804 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
rep Replicase polyprotein 1ab (378 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID

Mechanisms of Action

Mechanism of ActionAction Typetarget IDTarget NameTarget TypeTarget OrganismBinding Site NameReferences

Names and Identifiers

Canonical SMILES CC(C)C1=CC=C(C=C1)C2=NC(=O)N(C3=C2C=C(C=C3)OCC#C)C(C)C
Isomeric SMILES CC(C)C1=CC=C(C=C1)C2=NC(=O)N(C3=C2C=C(C=C3)OCC#C)C(C)C
PubChem CID 10109178
Molecular Weight 360.45

Certificates

Certificate of Analysis(COA)

Enter Lot Number to search for COA:

Chemical and Physical Properties

SolubilityDMSO : ≥ 100 mg/mL (277.43 mM)

Related Documents

Solution Calculators