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Regulators of G protein Signaling (RGS) proteins
CCG-203920 , CAS No.C608355, Inhibitor of regulator of G-protein signaling 4;Inhibitor of regulator of G-protein signaling 8

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CCG-203920 , CAS No.C608355, Inhibitor of regulator of G-protein signaling 4;Inhibitor of regulator of G-protein signaling 8

Moligand™

PubChem CID: 57330144

Item Number

C608355

Grouped product items
SKU	Size	Availability	Price	Qty
C608355-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,334.90
C608355-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90

View related series

regulator of G-protein signaling 4 Inhibitor regulator of G-protein signaling 8 Inhibitor

Basic Description

Synonyms	CCG203920;RGS4 inhibitor 13
Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	INHIBITOR
Mechanism of action	Inhibitor of regulator of G-protein signaling 4;Inhibitor of regulator of G-protein signaling 8

Associated Targets(Human)

RGS8 Tchem Regulator of G-protein signaling 8 (1 Activities)

Discover Target: RGS8

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

RGS4 Tchem Regulator of G-protein signaling 4 (2 Activities)

Discover Target: RGS4

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

CHRM3 Tclin Muscarinic acetylcholine receptor M3 (7750 Activities)

Discover Target: CHRM3

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

RGS4 Tchem Regulator of G-protein signaling 4 (13867 Activities)

Discover Target: RGS4

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

RGS8 Tchem Regulator of G-protein signaling 8 (45 Activities)

Discover Target: RGS8

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Names and Identifiers

IUPAC Name	2-ethyl-4-(2-methoxyethyl)-1,2,4-thiadiazolidine-3,5-dione
INCHI	InChI=1S/C7H12N2O3S/c1-3-9-6(10)8(4-5-12-2)7(11)13-9/h3-5H2,1-2H3
InChi Key	NCTIMJFWDQCLDW-UHFFFAOYSA-N
Canonical SMILES	COCCn1c(=O)sn(c1=O)CC
Isomeric SMILES	CCN1C(=O)N(C(=O)S1)CCOC
PubChem CID	57330144

Database links

PubChem CID	57330144
ChEMBL Ligand	CHEMBL2037369

Certificates

Certificate of Analysis(COA)

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References

1. Turner EM, Blazer LL, Neubig RR, Husbands SM. (2012) Small Molecule Inhibitors of Regulator of G Protein Signalling (RGS) Proteins.. ACS Med Chem Lett, 3 (2): (146-150). [PMID:22368763]

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