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Regulators of G protein Signaling (RGS) proteins
CCG-203920 , CAS No.C608355, Inhibitor of regulator of G-protein signaling 4;Inhibitor of regulator of G-protein signaling 8

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CCG-203920 , CAS No.C608355, Inhibitor of regulator of G-protein signaling 4;Inhibitor of regulator of G-protein signaling 8

Moligand™

PubChem CID: 57330144

Item Number

C608355

Grouped product items
SKU	Size	Availability	Price	Qty
C608355-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,334.90
C608355-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90

View related series

regulator of G-protein signaling 4 Inhibitor regulator of G-protein signaling 8 Inhibitor

Basic Description

Synonyms	CCG203920;RGS4 inhibitor 13
Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	INHIBITOR
Mechanism of action	Inhibitor of regulator of G-protein signaling 4;Inhibitor of regulator of G-protein signaling 8

Associated Targets(Human)

RGS8 Tchem Regulator of G-protein signaling 8 (1 Activities)

Discover Target: RGS8

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

RGS4 Tchem Regulator of G-protein signaling 4 (2 Activities)

Discover Target: RGS4

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

CHRM3 Tclin Muscarinic acetylcholine receptor M3 (7750 Activities)

Discover Target: CHRM3

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

RGS4 Tchem Regulator of G-protein signaling 4 (13867 Activities)

Discover Target: RGS4

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Mechanisms of Action

Mechanism of Action	Action Type	target ID	Target Name	Target Type	Target Organism	Binding Site Name	References

Names and Identifiers

IUPAC Name	2-ethyl-4-(2-methoxyethyl)-1,2,4-thiadiazolidine-3,5-dione
INCHI	InChI=1S/C7H12N2O3S/c1-3-9-6(10)8(4-5-12-2)7(11)13-9/h3-5H2,1-2H3
InChi Key	NCTIMJFWDQCLDW-UHFFFAOYSA-N
Canonical SMILES	COCCn1c(=O)sn(c1=O)CC
Isomeric SMILES	CCN1C(=O)N(C(=O)S1)CCOC
PubChem CID	57330144

Database links

PubChem CID	57330144
ChEMBL Ligand	CHEMBL2037369

Certificates

Certificate of Analysis(COA)

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References

1. Turner EM, Blazer LL, Neubig RR, Husbands SM. (2012) Small Molecule Inhibitors of Regulator of G Protein Signalling (RGS) Proteins.. ACS Med Chem Lett, 3 (2): (146-150). [PMID:22368763] [10.1021/op500134e]

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