JavaScript seems to be disabled in your browser. For the best experience on our site, be sure to turn on Javascript in your browser.

྾

CCG-4986 , CAS No.7134-19-2, Inhibitor of regulator of G-protein signaling 4

Item Number

C608358

Grouped product items
SKU	Size	Availability	Price	Qty
C608358-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$400.90
C608358-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,200.90

View related series

Basic Description

Synonyms	CCG-4986
Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	INHIBITOR
Mechanism of action	Inhibitor of regulator of G-protein signaling 4

RGS4 Tchem Regulator of G-protein signaling 4 (0 Activities)

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

IUPAC Name	(NE)-4-chloro-N-[methoxy-(4-nitrophenyl)-$l^{4}-sulfanylidene]benzenesulfonamide
INCHI	InChI=1S/C13H11ClN2O5S2/c1-21-22(12-6-4-11(5-7-12)16(17)18)15-23(19,20)13-8-2-10(14)3-9-13/h2-9H,1H3
InChi Key	GIFNUYPIOIDEGE-UHFFFAOYSA-N
Canonical SMILES	CO/S(=N/S(=O)(=O)c1ccc(cc1)Cl)/c1ccc(cc1)[N+](=O)[O-]
Isomeric SMILES	CO/S(=N/S(=O)(=O)C1=CC=C(C=C1)Cl)/C2=CC=C(C=C2)[N+](=O)[O-]
PubChem CID	5506256

PubChem CID	5506256
CAS Registry No.	7134-19-2

Enter Lot Number to search for COA:

1. Roman DL, Talbot JN, Roof RA, Sunahara RK, Traynor JR, Neubig RR. (2007) Identification of small-molecule inhibitors of RGS4 using a high-throughput flow cytometry protein interaction assay.. Mol Pharmacol, 71 (1): (169-75). [PMID:17012620] [10.1021/op500134e]
2. Roman DL, Blazer LL, Monroy CA, Neubig RR. (2010) Allosteric inhibition of the regulator of G protein signaling-Galpha protein-protein interaction by CCG-4986.. Mol Pharmacol, 78 (3): (360-5). [PMID:20530129] [10.1021/op500134e]

Determine the necessary mass, volume, or concentration for preparing a solution.

Determine the dilution needed to prepare a stock solution.