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Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
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SKU | Size | Availability | Price | Qty |
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C286617-2mg | 2mg | In stock | $62.90 | |
C286617-5mg | 5mg | In stock | $129.90 | |
C286617-10mg | 10mg | In stock | $195.90 | |
C286617-25mg | 25mg | In stock | $441.90 | |
C286617-50mg | 50mg | In stock | $783.90 | |
C286617-100mg | 100mg | In stock | $1,360.90 |
Highly selective and potent non-peptide NPY Y5receptor antagonist
Synonyms | AKOS024456984 | CGP 71683A; CGP71683A; CGP-71683 HCl | Q27258822 | MFCD00048633 | cgp71683a hcl | CGP-71683A HCl | N-[[4-[[(4-aminoquinazolin-2-yl)amino]methyl]cyclohexyl]methyl]naphthalene-1-sulfonamide;hydrochloride | SCHEMBL28512 | 45B73P82A3 | N-(((1r |
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Specifications & Purity | ≥99%(HPLC) |
Biochemical and Physiological Mechanisms | Extremely selective, non-peptide NPY Y5receptor antagonist. Displays > 1000-fold selectivity over Y1, Y2and Y4receptors; IC50values are 1.4, 2765, 7187 and 5637 nM at cloned rat Y5, Y1, Y2and Y4receptors respectively. Potently inhibits NPY-induced food in |
Storage Temp | Store at 2-8°C,Desiccated |
Shipped In | Wet ice |
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
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Mechanism of Action | Action Type | target ID | Target Name | Target Type | Target Organism | Binding Site Name | References |
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Pubchem Sid | 488196361 |
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Pubchem Sid Url | https://pubchem.ncbi.nlm.nih.gov/substance/488196361 |
IUPAC Name | N-[[4-[[(4-aminoquinazolin-2-yl)amino]methyl]cyclohexyl]methyl]naphthalene-1-sulfonamide;hydrochloride |
INCHI | InChI=1S/C26H29N5O2S.ClH/c27-25-22-9-3-4-10-23(22)30-26(31-25)28-16-18-12-14-19(15-13-18)17-29-34(32,33)24-11-5-7-20-6-1-2-8-21(20)24;/h1-11,18-19,29H,12-17H2,(H3,27,28,30,31);1H |
InChi Key | DIQDKUNCSVFGHH-UHFFFAOYSA-N |
Canonical SMILES | C1CC(CCC1CNC2=NC3=CC=CC=C3C(=N2)N)CNS(=O)(=O)C4=CC=CC5=CC=CC=C54.Cl |
Isomeric SMILES | C1CC(CCC1CNC2=NC3=CC=CC=C3C(=N2)N)CNS(=O)(=O)C4=CC=CC5=CC=CC=C54.Cl |
PubChem CID | 9849276 |
Molecular Weight | 512.07 |
Enter Lot Number to search for COA:
Find and download the COA for your product by matching the lot number on the packaging.
Lot Number | Certificate Type | Date | Item |
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E23161260 | Certificate of Analysis | Mar 30, 2023 | C286617 |
E2316376 | Certificate of Analysis | Mar 30, 2023 | C286617 |
E2316381 | Certificate of Analysis | Mar 30, 2023 | C286617 |
E2316385 | Certificate of Analysis | Mar 30, 2023 | C286617 |
E2316396 | Certificate of Analysis | Mar 30, 2023 | C286617 |
E2316402 | Certificate of Analysis | Mar 30, 2023 | C286617 |
E2316403 | Certificate of Analysis | Mar 30, 2023 | C286617 |
E2316404 | Certificate of Analysis | Mar 30, 2023 | C286617 |
E2316408 | Certificate of Analysis | Mar 30, 2023 | C286617 |
E2316409 | Certificate of Analysis | Mar 30, 2023 | C286617 |
E2316410 | Certificate of Analysis | Mar 30, 2023 | C286617 |
E2316412 | Certificate of Analysis | Mar 30, 2023 | C286617 |
Solubility | Solvent:DMSO, Max Conc. mg/mL: 51.21, Max Conc. mM: 100 |
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Starting at $241.90