CGP 71683 hydrochloride - 10mM in DMSO, high purity , CAS No.192322-50-2

  • 10mM in DMSO
Item Number
C422353
Grouped product items
SKUSizeAvailabilityPrice Qty
C422353-1ml
1ml
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$241.90

Highly selective and potent non-peptide NPY Y5receptor antagonist

Basic Description

SynonymsAKOS024456984 | CGP 71683A; CGP71683A; CGP-71683 HCl | Q27258822 | MFCD00048633 | cgp71683a hcl | CGP-71683A HCl | N-[[4-[[(4-aminoquinazolin-2-yl)amino]methyl]cyclohexyl]methyl]naphthalene-1-sulfonamide;hydrochloride | SCHEMBL28512 | 45B73P82A3 | N-(((1r
Specifications & Purity10mM in DMSO
Biochemical and Physiological MechanismsExtremely selective, non-peptide NPY Y5receptor antagonist. Displays > 1000-fold selectivity over Y1, Y2and Y4receptors; IC50values are 1.4, 2765, 7187 and 5637 nM at cloned rat Y5, Y1, Y2and Y4receptors respectively. Potently inhibits NPY-induced food in
Storage TempStore at -80°C
Shipped InIce chest + Ice pads

Associated Targets(non-human)

Plasmodium falciparum (966862 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID

Mechanisms of Action

Mechanism of ActionAction Typetarget IDTarget NameTarget TypeTarget OrganismBinding Site NameReferences

Names and Identifiers

IUPAC Name N-[[4-[[(4-aminoquinazolin-2-yl)amino]methyl]cyclohexyl]methyl]naphthalene-1-sulfonamide;hydrochloride
INCHI InChI=1S/C26H29N5O2S.ClH/c27-25-22-9-3-4-10-23(22)30-26(31-25)28-16-18-12-14-19(15-13-18)17-29-34(32,33)24-11-5-7-20-6-1-2-8-21(20)24;/h1-11,18-19,29H,12-17H2,(H3,27,28,30,31);1H
InChi Key DIQDKUNCSVFGHH-UHFFFAOYSA-N
Canonical SMILES C1CC(CCC1CNC2=NC3=CC=CC=C3C(=N2)N)CNS(=O)(=O)C4=CC=CC5=CC=CC=C54.Cl
Isomeric SMILES C1CC(CCC1CNC2=NC3=CC=CC=C3C(=N2)N)CNS(=O)(=O)C4=CC=CC5=CC=CC=C54.Cl
PubChem CID 9849276
Molecular Weight 512.07

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