cipralisant , CAS No.213027-19-1, Agonist of H 3 receptor

Item Number

C608570

Grouped product items
SKU	Size	Availability	Price	Qty
C608570-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,258.90
C608570-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$4,000.90

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Basic Description

Synonyms	CIPRALISANT \| Cipralisant [INN] \| 213027-19-1 \| GT-2331 \| Cipralisant, (-)- \| 309713XSKW \| UNII-309713XSKW \| CHEMBL278462 \| 5-[(1R,2R)-2-(5,5-dimethylhex-1-ynyl)cyclopropyl]-1H-imidazole \| (-)-GT-2331 \| 4-((1R,2R)-2-(5,5-Dimethylhex-1-ynyl)cyclopropyl)-1H-imidazole \| GTPL1244 \|
Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	AGONIST
Mechanism of action	Agonist of H 3 receptor

Associated Targets(Human)

HRH3 Tclin Histamine H3 receptor (4 Activities)

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

HRH3 Tclin Histamine H3 receptor (10389 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Names and Identifiers

IUPAC Name	5-[(1R,2R)-2-(5,5-dimethylhex-1-ynyl)cyclopropyl]-1H-imidazole
INCHI	InChI=1S/C14H20N2/c1-14(2,3)7-5-4-6-11-8-12(11)13-9-15-10-16-13/h9-12H,5,7-8H2,1-3H3,(H,15,16)/t11-,12-/m1/s1
InChi Key	CVKJAXCQPFOAIN-VXGBXAGGSA-N
Canonical SMILES	CC(C)(C)CCC#CC1CC1C2=CN=CN2
Isomeric SMILES	CC(C)(C)CCC#C[C@@H]1C[C@H]1C2=CN=CN2
Alternate CAS	213027-19-1
PubChem CID	6450823
MeSH Entry Terms	4-(2-(5,5-dimethylhex-1-ynyl)cyclopropyl)imidazole;GT 2331;GT-2331

PubChem CID

Wikipedia

CAS Registry No.

ChEMBL Ligand

GPCRdb Ligand

References

1. Krueger KM, Witte DG, Ireland-Denny L, Miller TR, Baranowski JL, Buckner S, Milicic I, Esbenshade TA, Hancock AA. (2005) G protein-dependent pharmacology of histamine H3 receptor ligands: evidence for heterogeneous active state receptor conformations.. J Pharmacol Exp Ther, 314 (1): (271-81). [PMID:15821027]

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Basic Description