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Cisapride - ≥99%, high purity , CAS No.81098-60-4, Agonist of 5-HT 4 receptor;Agonist of 5-HT 7 receptor;Channel blocker of K v11.1
5-HT 4 receptor agonist. hERG blocker.
Basic Description Synonyms R-51619 | SCHEMBL16132 | SR-01000597514-1 | cis-4-amino-5-chloro-N-(1-(3-(p-fluorophenoxy)propyl)-3-methoxy-4-piperidinyl)-o-anisamide | Pridesia | 4-amino-5-chloro-N-(cis-1-(3-(4-fluorophenoxy)propyl)-3-methoxypiperidin-4-yl)-2-methoxybenzamide | Acpulsi Specifications & Purity Moligand™, ≥99% Biochemical and Physiological Mechanisms 5-HT 4 receptor agonist (EC 50 = 140 nM). Potent human ether-a-go-go-related gene (hERG) channel blocker (IC 50 = 9.4 nM). Gastrokinetic agent, increases intestinal motility. Storage Temp Store at -20°C Shipped In Ice chest + Ice pads Grade Moligand™ Action Type AGONIST, CHANNEL BLOCKER Mechanism of action Agonist of 5-HT 4 receptor;Agonist of 5-HT 7 receptor;Channel blocker of K v11.1 Note Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details. Product Description Product Description：
Associated Targets(Human) Associated Targets(non-human) Mechanisms of Action Mechanism of Action Action Type target ID Target Name Target Type Target Organism Binding Site Name References
Names and Identifiers IUPAC Name 4-amino-5-chloro-N-[(3S,4R)-1-[3-(4-fluorophenoxy)propyl]-3-methoxypiperidin-4-yl]-2-methoxybenzamide INCHI InChI=1S/C23H29ClFN3O4/c1-30-21-13-19(26)18(24)12-17(21)23(29)27-20-8-10-28(14-22(20)31-2)9-3-11-32-16-6-4-15(25)5-7-16/h4-7,12-13,20,22H,3,8-11,14,26H2,1-2H3,(H,27,29)/t20-,22+/m1/s1 InChi Key DCSUBABJRXZOMT-IRLDBZIGSA-N Canonical SMILES COC1CN(CCC1NC(=O)C2=CC(=C(C=C2OC)N)Cl)CCCOC3=CC=C(C=C3)F Isomeric SMILES CO[C@H]1CN(CC[C@H]1NC(=O)C2=CC(=C(C=C2OC)N)Cl)CCCOC3=CC=C(C=C3)F PubChem CID 6917698 Molecular Weight 465.95
Chemical and Physical Properties Solubility Soluble in DMSO to 100 mM and in ethanol to 25 mM (with warming)
Safety and Hazards(GHS) Pictogram(s) GHS05 Signal Danger Hazard Statements H318: Causes serious eye damage
Precautionary Statements P280: Wear protective gloves/protective clothing/eye protection/face protection.
P264+P265: Wash hands [and …] thoroughly after handling. Do not touch eyes.
P305+P354+P338: IF IN EYES: Immediately rinse with water for several minutes. Remove contact lenses if present and easy to do. Continue rinsing.
P317: Get emergency medical help.
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K2103559