Cisapride - ≥99%, high purity , CAS No.81098-60-4, Agonist of 5-HT 4 receptor;Agonist of 5-HT 7 receptor;Channel blocker of K v11.1

Item Number

C275070

• Synonyms: R-51619 | SCHEMBL16132 | SR-01000597514-1 | cis-4-amino-5-chloro-N-(1-(3-(p-fluorophenoxy)propyl)-3-methoxy-4-piperidinyl)-o-anisamide | Pridesia | 4-amino-5-chloro-N-(cis-1-(3-(4-fluorophenoxy)propyl)-3-methoxypiperidin-4-yl)-2-methoxybenzamide | Acpulsi
• Specifications & Purity: Moligand™, ≥99%
• Biochemical and Physiological Mechanisms: 5-HT 4 receptor agonist (EC 50 = 140 nM). Potent human ether-a-go-go-related gene (hERG) channel blocker (IC 50 = 9.4 nM). Gastrokinetic agent, increases intestinal motility.
• Storage Temp: Store at -20°C
• Shipped In: Ice chest + Ice pads
• Grade: Moligand™
• Action Type: AGONIST, CHANNEL BLOCKER
• Mechanism of action: Agonist of 5-HT 4 receptor;Agonist of 5-HT 7 receptor;Channel blocker of K v11.1
• Note: Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.

Product Description

Product Description：
Cisapride (R 51619, Kaudalit, Kinestase, Prepulsid, Presid, Pridesia, Propulsid) is a nonselective 5-HT4 receptor agonist with gastroprokinetic effects.