Skip to the beginning of the images gallery

Cisapride - ≥99%, high purity , CAS No.81098-60-4, Agonist of 5-HT 4 receptor;Agonist of 5-HT 7 receptor;Channel blocker of K v11.1

Moligand™
≥99%

CAS#: 81098-60-4
Formula: C₂₃H₂₉ClFN₃O₄
Molecular Weight: 465.95
PubChem CID: 6917698

Item Number

C275070

Grouped product items
SKU	Size	Availability	Price
C275070-10mg	10mg	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$77.90
C275070-50mg	50mg	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$122.90
C275070-100mg	100mg	In stock	$195.90
C275070-250mg	250mg	In stock	$441.90

5-HT 4 receptor agonist. hERG blocker.

View related series

5-HT4 receptor Agonist 5-HT7 receptor Agonist Kv11.1 Channel blocker

Basic Description

Synonyms	cisapride\|81098-60-4\|Cisaprida\|Cisapridum\|Prepulsid\|Kaudalit\|Pridesia\|(+-)-Cisapride\|CHEBI:3720\|R 51619\|Propulsid\|Acenalin\|Risamol\|UVL329170W\|86718-70-9\|Kinestase\|cis-4-Amino-5-chloro-N-(1-(3-(p-fluorophenoxy)propyl)-3-methoxy-4-piperidyl)-o-anisamide\|CHE
Specifications & Purity	≥99%
Storage Temp	Store at -20°C
Shipped In	Dry ice
Grade	Moligand™
Action Type	AGONIST, CHANNEL BLOCKER
Mechanism of action	Agonist of 5-HT 4 receptor;Agonist of 5-HT 7 receptor;Channel blocker of K v11.1
Product Description	Product Description： Cisapride (R 51619, Kaudalit, Kinestase, Prepulsid, Presid, Pridesia, Propulsid) is a nonselective 5-HT4 receptor agonist with gastroprokinetic effects.

Associated Targets

HTR4 Tclin 5-hydroxytryptamine receptor 4 1 Activities

Discover Target: HTR4

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

HTR7 Tclin 5-hydroxytryptamine receptor 7 1 Activities

Discover Target: HTR7

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

KCNH2 Tclin Potassium voltage-gated channel subfamily H member 2 2 Activities

Discover Target: KCNH2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	4-amino-5-chloro-N-[(3S,4R)-1-[3-(4-fluorophenoxy)propyl]-3-methoxypiperidin-4-yl]-2-methoxybenzamide
INCHI	InChI=1S/C23H29ClFN3O4/c1-30-21-13-19(26)18(24)12-17(21)23(29)27-20-8-10-28(14-22(20)31-2)9-3-11-32-16-6-4-15(25)5-7-16/h4-7,12-13,20,22H,3,8-11,14,26H2,1-2H3,(H,27,29)/t20-,22+/m1/s1
InChi Key	DCSUBABJRXZOMT-IRLDBZIGSA-N
Canonical SMILES	COC1CN(CCC1NC(=O)C2=CC(=C(C=C2OC)N)Cl)CCCOC3=CC=C(C=C3)F
Isomeric SMILES	CO[C@H]1CN(CC[C@H]1NC(=O)C2=CC(=C(C=C2OC)N)Cl)CCCOC3=CC=C(C=C3)F
PubChem CID	6917698
Molecular Weight	465.95

PubChem CID

ChEBI

Wikipedia

ChEMBL Ligand

DrugBank Ligand

BindingDB Ligand

CAS Registry No.

DrugCentral Ligand

GPCRdb Ligand

Certificates

Certificate of Analysis(COA)

Enter Lot Number to search for COA:

To view the certificate results,please click on a Lot number.For Lot numbers from past orders,please use our order status section

4 results found

Lot Number	Certificate Type	Date	Item
K2103559	Certificate of Analysis	Jun 14, 2023	C275070
K2103561	Certificate of Analysis	Jun 14, 2023	C275070
K2103790	Certificate of Analysis	Jun 14, 2023	C275070
K2103791	Certificate of Analysis	Jun 14, 2023	C275070

Safety and Hazards(GHS)

Pictogram(s)	GHS05
Signal	Danger
Hazard Statements	H318:Causes serious eye damage
Precautionary Statements	P280:Wear protective gloves/protective clothing/eye protection/face protection. P264+P265:Wash hands [and …] thoroughly after handling. Do not touch eyes. P305+P354+P338:IF IN EYES: Immediately rinse with water for several minutes. Remove contact lenses if present and easy to do. Continue rinsing. P317:Get emergency medical help.

Solution Calculators

Molarity Calculator

Determine the necessary mass, volume, or concentration for preparing a solution.

Dilution Calculator

Determine the dilution needed to prepare a stock solution.