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[d-Tyr-¹⁴C]TAK-448 , CAS No.D610007, Agonist of kisspeptin receptor

Item Number

D610007

Grouped product items
SKU	Size	Availability	Price	Qty
D610007-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,400.90
D610007-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90

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Basic Description

Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	AGONIST
Mechanism of action	Agonist of kisspeptin receptor

KISS1R Tchem KiSS-1 receptor (0 Activities)

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

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1. Nishizawa N, Takatsu Y, Kumano S, Kiba A, Ban J, Tsutsumi S, Matsui H, Matsumoto SI, Yamaguchi M, Ikeda Y et al.. (2016) Design and Synthesis of an Investigational Nonapeptide KISS1 Receptor (KISS1R) Agonist, Ac-d-Tyr-Hydroxyproline (Hyp)-Asn-Thr-Phe-azaGly-Leu-Arg(Me)-Trp-NH₂ (TAK-448), with Highly Potent Testosterone-Suppressive Activity and Excellent Water Solubility.. J Med Chem, 59 (19): (8804-8811). [PMID:27589480] [10.1021/op500134e]
2. Moriya Y, Kogame A, Tagawa Y, Morohashi A, Kondo T, Asahi S. (2019) Investigation of disposition for TAK-448, a synthetic peptide of kisspeptin analog, in rats and dogs using the radiolabeled TAK-448 suitable for pharmacokinetic study.. Xenobiotica, 49 (7): (833-839). [PMID:30044673] [10.1021/op500134e]

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