Standard InChI: InChI=1S/C17H28N8O5/c1-20-3-5-24(4-2-9(18)17(28)29)6-10-12(26)13(27)16(30-10)25-8-23-11-14(19)21-7-22-15(11)25/h7-10,12-13,16,20,26-27H,2-6,18H2,1H3,(H,28,29)(H2,19,21,22)/t9-,10+,12+,13+,16+/m0/s1
1.Mori S, Iwase K, Iwanami N, Tanaka Y, Kagechika H, Hirano T.. (2010) Development of novel bisubstrate-type inhibitors of histone methyltransferase SET7/9., 18 (23):[PMID:21036620][10.1016/j.bmc.2010.10.022]
2.Barsyte-Lovejoy, Dalia D and 32 more authors. 2014-09-02 (R)-PFI-2 is a potent and selective inhibitor of SETD7 methyltransferase activity in cells. [PMID:25136132]
3.Kaniskan, H Ümit; Konze, Kyle D and Jin, Jian. 2015-02-26 Selective inhibitors of protein methyltransferases. [PMID:25406853]
4.Takemoto, Yasushi Y and 16 more authors. 2016-04-28 Identification of Cyproheptadine as an Inhibitor of SET Domain Containing Lysine Methyltransferase 7/9 (Set7/9) That Regulates Estrogen-Dependent Transcription. [PMID:27088648]
5.Min, Wenjian and 10 more authors. 2020-04-01 Computational discovery and biological evaluation of novel inhibitors targeting histone-lysine N-methyltransferase SET7. [PMID:32088124]